Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004252 | molecular_function | serine-type endopeptidase activity |
A | 0005615 | cellular_component | extracellular space |
A | 0005737 | cellular_component | cytoplasm |
A | 0006508 | biological_process | proteolysis |
A | 0008236 | molecular_function | serine-type peptidase activity |
A | 0043231 | cellular_component | intracellular membrane-bounded organelle |
B | 0004252 | molecular_function | serine-type endopeptidase activity |
B | 0005615 | cellular_component | extracellular space |
B | 0005737 | cellular_component | cytoplasm |
B | 0006508 | biological_process | proteolysis |
B | 0008236 | molecular_function | serine-type peptidase activity |
B | 0043231 | cellular_component | intracellular membrane-bounded organelle |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE SO4 A 246 |
Chain | Residue |
A | ARG161 |
A | ASN185 |
A | LYS186 |
A | ARG188 |
A | HOH265 |
B | LYS93 |
site_id | AC2 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE SO4 A 247 |
Chain | Residue |
A | ALA204 |
A | GLY205 |
A | HOH258 |
B | ARG49 |
A | ARG27 |
A | ARG137 |
A | LEU200 |
site_id | AC3 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE SO4 B 246 |
Chain | Residue |
A | LYS87 |
B | ARG161 |
B | ASN185 |
B | LYS186 |
B | ARG188 |
B | HOH249 |
site_id | AC4 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE SO4 B 247 |
Chain | Residue |
B | ARG27 |
B | ARG137 |
B | LEU200 |
B | ALA204 |
B | GLY205 |
B | HOH269 |
site_id | AC5 |
Number of Residues | 15 |
Details | BINDING SITE FOR CHAIN I OF METHOXYSUCCINYL-ALA-ALA-PRO-ALA CHLOROMETHYL KETONE INHIBITOR |
Chain | Residue |
A | HIS57 |
A | TYR191 |
A | GLY193 |
A | SER195 |
A | SER214 |
A | TYR215 |
A | VAL216 |
A | LEU217 |
A | ARG218 |
A | ASN219 |
A | HOH284 |
B | PRO185 |
B | LYS186 |
B | ILE187 |
I | HOH7 |
site_id | AC6 |
Number of Residues | 11 |
Details | BINDING SITE FOR CHAIN J OF METHOXYSUCCINYL-ALA-ALA-PRO-ALA CHLOROMETHYL KETONE INHIBITOR |
Chain | Residue |
A | HOH279 |
B | HIS57 |
B | TYR191 |
B | GLY193 |
B | SER195 |
B | SER214 |
B | TYR215 |
B | VAL216 |
B | ARG218 |
B | ASN219 |
J | HOH7 |
Functional Information from PROSITE/UniProt
site_id | PS00134 |
Number of Residues | 6 |
Details | TRYPSIN_HIS Serine proteases, trypsin family, histidine active site. MTAAHC |
Chain | Residue | Details |
A | MET53-CYS58 | |
site_id | PS00135 |
Number of Residues | 12 |
Details | TRYPSIN_SER Serine proteases, trypsin family, serine active site. NVykGDSGGPLL |
Chain | Residue | Details |
A | ASN189-LEU200 | |