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2Q6M

Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with the PJ34 inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0047286molecular_functionNAD+-diphthamide ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE P34 A 1001
ChainResidue
AHIS460
AGLY461
ATYR493
AALA501
ATYR504
AGLU581
AHOH1190

site_idAC2
Number of Residues13
DetailsBINDING SITE FOR RESIDUE P34 A 1002
ChainResidue
AGLU452
ATYR454
AASN550
AALA576
AHIS591
AALA592
AVAL593
AHOH1068
AHOH1223
AHOH1247
AHOH1342
ATHR445
ALEU449

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000305
ChainResidueDetails
AGLU581

Catalytic Information from CSA
site_idCSA1
Number of Residues1
DetailsAnnotated By Reference To The Literature 1zm2
ChainResidueDetails
AGLU581

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PDB entries from 2024-07-17

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