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2OUO

Crystal Structure of the Bromo domain 2 in human Bromodomain Containing Protein 4 (BRD4)

Functional Information from PDB Data
site_idAC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 201
ChainResidue
AHOH11
AASN433

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 202
ChainResidue
AHOH84
AHOH158
ALEU424
ASER427
AASN428
ALYS431
AALA455

site_idAC3
Number of Residues1
DetailsBINDING SITE FOR RESIDUE EDO A 203
ChainResidue
AGLU438

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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