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2MW6

Structure of the bee venom toxin melittin with [(C5H5)Ru]+ fragment attached to the tryptophan residue

Functional Information from GO Data
ChainGOidnamespacecontents
A0004860molecular_functionprotein kinase inhibitor activity
A0005576cellular_componentextracellular region
Functional Information from PDB Data
site_idAC1
Number of Residues1
DetailsBINDING SITE FOR RESIDUE 3UQ A 101
ChainResidue
ATRP19

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues25
DetailsPeptide: {"description":"Melittin","featureId":"PRO_0000035149","evidences":[{"source":"PubMed","id":"20403370","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"20472009","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"5592400","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Important for the flexibility at the center of the helix, flexibility that is important for the stability of the voltage-gated pore","evidences":[{"source":"PubMed","id":"2187536","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsModified residue: {"description":"N-formylglycine; partial","evidences":[{"source":"PubMed","id":"5139483","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues1
DetailsModified residue: {"description":"Glutamine amide","evidences":[{"source":"PubMed","id":"5592400","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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