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2JJJ

Endothiapepsin in complex with a gem-diol inhibitor.

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues23
DetailsBINDING SITE FOR RESIDUE 0QS A 331
ChainResidue
AASP15
APHE116
AASP119
ALEU133
AASP219
AGLY221
ATHR222
ATHR223
AILE300
AILE304
AHOH2260
AASP33
AHOH2398
AHOH2518
AHOH2519
AHOH2520
AASP35
AGLY37
ASER38
ATYR79
AGLY80
AASP81
ASER83

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE SO4 A 500
ChainResidue
ASER113
ASER114
ATHR321
ATHR322
ASO4503
AHOH2237
AHOH2507
AHOH2508
AHOH2509
AHOH2510

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 501
ChainResidue
ALYS68
ALEU69
AHOH2511
AHOH2512

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 502
ChainResidue
ALYS191
AHOH2513
AHOH2515

site_idAC5
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 503
ChainResidue
AASP81
AGLY82
ASER83
ASER113
ASER114
ASER115
ASO4500
AHOH2516
AHOH2517

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. LDFDTGSSDLWV
ChainResidueDetails
ALEU32-VAL43
AILE217-PRO228

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE:
ChainResidueDetails
AASP35
ATHR200

Catalytic Information from CSA
site_idCSA1
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
ASER38
AASP35
ATHR222
AASP219

site_idCSA2
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP35
ATHR220
AASP219
ATHR36

site_idCSA3
Number of Residues3
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
ASER38
AASP35
AASP219

site_idCSA4
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP35
ATHR222
AASP219
ATHR36

site_idCSA5
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP35

site_idCSA6
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP219

237735

PDB entries from 2025-06-18

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