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2HUW

X-ray crystal structure of the Grb2 SH2 domain complexed to a constrained and cyclopropane-derived ligand

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 B 201
ChainResidue
BHIS58
BPRO59
BTRP60
BARG136
BASP150
BHOH220

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE YVN B 202
ChainResidue
BSER88
BGLU89
BSER90
BSER96
BHIS107
BPHE108
BLYS109
BLEU120
BTRP121
BHOH228
BHOH246
BHOH250
BHOH268
APRO155
BARG67
BARG86

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE YVN A 203
ChainResidue
AARG67
AARG86
ASER88
AGLU89
ASER90
ASER96
AGLN106
AHIS107
APHE108
ALYS109
ALEU120
ATRP121
AHOH223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861
ChainResidueDetails
ALYS109
BLYS109

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PDB entries from 2024-07-24

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