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2GPP

Estrogen Related Receptor-gamma ligand binding domain complexed with a RIP140 peptide and synthetic ligand GSK4716

Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 1BA A 459
ChainResidue
AHOH1
AVAL313
AARG316
AVAL325
ATYR326
AASP328
AHOH23
AGLU247
ALYS248
AILE249
ALEU268
AALA272
AGLU275
ALEU309

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues224
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 5"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"UniProtKB","id":"Q8CBD1","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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