Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE K E 247 |
| Chain | Residue |
| E | GLU128 |
| E | SER130 |
| F | GLU128 |
| F | SER130 |
| site_id | AC2 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE K D 247 |
| Chain | Residue |
| C | GLU128 |
| C | SER130 |
| D | GLU128 |
| D | SER130 |
| site_id | AC3 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE K G 247 |
| Chain | Residue |
| G | GLU128 |
| G | SER130 |
| G | SER130 |
| G | GLU128 |
| site_id | AC4 |
| Number of Residues | 1 |
| Details | BINDING SITE FOR RESIDUE K B 247 |
| site_id | AC5 |
| Number of Residues | 3 |
| Details | BINDING SITE FOR RESIDUE K B 248 |
| Chain | Residue |
| A | GLU128 |
| B | GLU128 |
| B | SER130 |
| site_id | AC6 |
| Number of Residues | 1 |
| Details | BINDING SITE FOR RESIDUE K F 247 |
| site_id | AC7 |
| Number of Residues | 1 |
| Details | BINDING SITE FOR RESIDUE K C 247 |
| site_id | AC8 |
| Number of Residues | 1 |
| Details | BINDING SITE FOR RESIDUE K D 248 |
| site_id | AC9 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO D 249 |
| Chain | Residue |
| D | TYR58 |
| D | TYR72 |
| D | LEU75 |
| D | MSE76 |
| D | ASP79 |
| D | TRP188 |
| site_id | BC1 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO B 249 |
| Chain | Residue |
| B | TYR58 |
| B | TYR72 |
| B | LEU75 |
| B | MSE76 |
| B | ASP79 |
| B | TRP188 |
| site_id | BC2 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO C 248 |
| Chain | Residue |
| C | TYR58 |
| C | TYR72 |
| C | LEU75 |
| C | MSE76 |
| C | ASP79 |
| C | TRP168 |
| C | TRP188 |
| site_id | BC3 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO G 248 |
| Chain | Residue |
| G | TYR58 |
| G | TYR72 |
| G | LEU75 |
| G | MSE76 |
| G | ASP79 |
| G | TRP188 |
| site_id | BC4 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO E 248 |
| Chain | Residue |
| E | TYR58 |
| E | TYR72 |
| E | LEU75 |
| E | MSE76 |
| E | ASP79 |
| E | TRP188 |
| E | EDO250 |
| site_id | BC5 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO A 247 |
| Chain | Residue |
| A | ARG10 |
| A | TYR116 |
| A | TRP191 |
| A | ASN192 |
| A | EDO248 |
| A | HOH422 |
| site_id | BC6 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO A 248 |
| Chain | Residue |
| A | TYR58 |
| A | TYR72 |
| A | LEU75 |
| A | MSE76 |
| A | ASP79 |
| A | TRP188 |
| A | EDO247 |
| site_id | BC7 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO G 249 |
| Chain | Residue |
| G | ASP79 |
| G | ILE138 |
| G | CYS164 |
| G | TRP168 |
| G | GLU229 |
| G | VAL232 |
| G | HOH382 |
| site_id | BC8 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO D 250 |
| Chain | Residue |
| D | ASP79 |
| D | TYR82 |
| D | ILE138 |
| D | CYS164 |
| D | TRP168 |
| D | GLU229 |
| D | HOH375 |
| site_id | BC9 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO B 250 |
| Chain | Residue |
| B | ASP79 |
| B | CYS164 |
| B | TRP168 |
| B | GLU229 |
| B | VAL232 |
| B | PHE233 |
| B | HOH378 |
| site_id | CC1 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO C 249 |
| Chain | Residue |
| C | ASP79 |
| C | ILE138 |
| C | CYS164 |
| C | TRP168 |
| C | GLU229 |
| C | VAL232 |
| C | HOH393 |
| site_id | CC2 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE EDO E 249 |
| Chain | Residue |
| E | ASP79 |
| E | TYR82 |
| E | TYR141 |
| E | GLU229 |
| E | VAL232 |
| E | PHE233 |
| E | HOH360 |
| site_id | CC3 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO A 249 |
| Chain | Residue |
| A | ASP79 |
| A | CYS164 |
| A | TRP168 |
| A | GLU229 |
| A | VAL232 |
| A | HOH364 |
| site_id | CC4 |
| Number of Residues | 8 |
| Details | BINDING SITE FOR RESIDUE EDO F 248 |
| Chain | Residue |
| F | ASP79 |
| F | TYR82 |
| F | CYS164 |
| F | TRP168 |
| F | GLU229 |
| F | VAL232 |
| F | PHE233 |
| F | HOH409 |
| site_id | CC5 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO E 250 |
| Chain | Residue |
| E | ARG10 |
| E | TYR116 |
| E | TRP191 |
| E | ASN192 |
| E | EDO248 |
| E | HOH433 |
| site_id | CC6 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO E 251 |
| Chain | Residue |
| E | ARG24 |
| E | LEU28 |
| E | THR101 |
| E | GLN208 |
| E | HOH475 |
| site_id | CC7 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO G 250 |
| Chain | Residue |
| G | ARG24 |
| G | THR27 |
| G | LEU28 |
| G | THR101 |
| G | GLN208 |
| site_id | CC8 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO A 250 |
| Chain | Residue |
| A | THR224 |
| A | ASN227 |
| A | TYR228 |
| A | LYS231 |
| A | HOH298 |
| G | GLU100 |
| site_id | CC9 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO F 249 |
| Chain | Residue |
| A | TYR178 |
| F | TYR178 |
| F | HOH420 |
| F | HOH451 |
| F | HOH454 |
| site_id | DC1 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO D 251 |
| Chain | Residue |
| C | THR224 |
| C | ASN227 |
| C | TYR228 |
| C | LYS231 |
| D | GLU100 |
| D | ARG103 |
| site_id | DC2 |
| Number of Residues | 3 |
| Details | BINDING SITE FOR RESIDUE EDO F 250 |
| Chain | Residue |
| F | ARG24 |
| F | LEU28 |
| F | GLN208 |
| site_id | DC3 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO D 252 |
| Chain | Residue |
| D | ARG24 |
| D | THR27 |
| D | LEU28 |
| D | GLN208 |
| D | HOH448 |
| site_id | DC4 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO C 250 |
| Chain | Residue |
| C | ARG24 |
| C | THR27 |
| C | LEU28 |
| C | THR101 |
| C | GLN208 |
| C | HOH390 |
| site_id | DC5 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE EDO G 251 |
| Chain | Residue |
| G | THR224 |
| G | ASN227 |
| G | TYR228 |
| G | LYS231 |
| site_id | DC6 |
| Number of Residues | 6 |
| Details | BINDING SITE FOR RESIDUE EDO F 251 |
| Chain | Residue |
| F | TYR58 |
| F | TYR72 |
| F | LEU75 |
| F | MSE76 |
| F | ASP79 |
| F | TRP188 |
| site_id | DC7 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE EDO E 252 |
| Chain | Residue |
| E | TYR166 |
| E | ASN173 |
| E | TYR200 |
| E | HOH340 |
| site_id | DC8 |
| Number of Residues | 5 |
| Details | BINDING SITE FOR RESIDUE EDO F 252 |
| Chain | Residue |
| C | THR22 |
| C | HOH319 |
| C | HOH374 |
| F | ASP137 |
| F | LYS231 |
| site_id | DC9 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE EDO A 251 |
| Chain | Residue |
| A | ASP31 |
| A | VAL32 |
| A | PRO33 |
| A | ASN204 |