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1XNX

Crystal structure of constitutive androstane receptor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE ATE A 500
ChainResidue
AHOH16
APHE171
AASN175
APHE227
ALYS235
AALA239
ALEU253

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ATE B 600
ChainResidue
BASN175
BPHE227
BHOH29
BPHE171

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsSite: {"description":"Important for TCPOBOP recognition"}
ChainResidueDetails

240971

PDB entries from 2025-08-27

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