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1QF2

THERMOLYSIN (E.C.3.4.24.27) COMPLEXED WITH (2-SULPHANYL-3-PHENYLPROPANOYL)-GLY-(5-PHENYLPROLINE). PARAMETERS FOR ZN-MONODENTATION OF MERCAPTOACYLDIPEPTIDES IN METALLOENDOPEPTIDASE

Functional Information from GO Data
ChainGOidnamespacecontents
A0004222molecular_functionmetalloendopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 320
ChainResidue
AHIS142
AHIS146
AGLU166
ATI3317

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 321
ChainResidue
AASP185
AGLU187
AGLU190
AHOH331
AASP138
AGLU177

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 322
ChainResidue
AGLU177
AASN183
AASP185
AGLU190
AHOH341
AHOH351

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 323
ChainResidue
AASP57
AASP59
AGLN61
AHOH328
AHOH352
AHOH381

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 324
ChainResidue
ATYR193
ATHR194
AILE197
AASP200
AHOH350
AHOH380

site_idAC6
Number of Residues14
DetailsBINDING SITE FOR RESIDUE TI3 A 317
ChainResidue
AASN111
AASN112
APHE130
ALEU133
AVAL139
AHIS142
AGLU143
AGLU166
ALEU202
AARG203
AHIS231
AZN320
AHOH492
AHOH543

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE DMS A 325
ChainResidue
ASER218
ATYR251

site_idAC8
Number of Residues2
DetailsBINDING SITE FOR RESIDUE DMS A 326
ChainResidue
ATRP115
AHIS146

site_idAC9
Number of Residues1
DetailsBINDING SITE FOR RESIDUE DMS A 327
ChainResidue
ATYR151

site_idZN
Number of Residues3
DetailsZN BINDING SITE
ChainResidue
AHIS146
AHIS142
AGLU166

Functional Information from PROSITE/UniProt
site_idPS00142
Number of Residues10
DetailsZINC_PROTEASE Neutral zinc metallopeptidases, zinc-binding region signature. VVAHELTHAV
ChainResidueDetails
AVAL139-VAL148

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING:
ChainResidueDetails
AVAL289
ASER291
ATHR293

Catalytic Information from CSA
site_idMCSA1
Number of Residues
DetailsM-CSA 176
ChainResidueDetails

218853

PDB entries from 2024-04-24

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