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1Q4X

Crystal Structure of Human Thyroid Hormone Receptor beta LBD in complex with specific agonist GC-24

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE G24 A 462
ChainResidue
APHE269
AHIS435
APHE451
APHE455
APHE272
ATHR273
AALA279
AARG316
AARG320
AASN331
AGLY332
ALEU346

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE G24 A 463
ChainResidue
AHOH25
ALEU365
AASP366
AVAL376
ASER380
ASER381
AGLU393
AGLN396
AARG429

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:15466465, ECO:0007744|PDB:1Y0X
ChainResidueDetails
AARG282
AASN331
AHIS435

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PDB entries from 2025-06-18

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