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1N46

CRYSTAL STRUCTURE OF HUMAN TR BETA LIGAND-BINDING DOMAIN COMPLEXED WITH A POTENT SUBTYPE-SELECTIVE THYROMIMETIC

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE PFA A 462
ChainResidue
APHE272
ALEU330
AASN331
AGLY344
ALEU346
AHIS435
AMET442
APHE455
AILE276
AALA279
AARG282
AMET310
AMET313
AARG316
AALA317
AARG320

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE PFA B 463
ChainResidue
BPHE272
BILE276
BALA279
BARG282
BMET310
BMET313
BARG316
BARG320
BASN331
BGLY344
BLEU346
BILE353
BHIS435
BMET442
BPHE455

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15466465, ECO:0007744|PDB:1Y0X
ChainResidueDetails
AARG282
AASN331
AHIS435
BARG282
BASN331
BHIS435

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PDB entries from 2024-07-17

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