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1KUG

Crystal Structure of a Taiwan Habu Venom Metalloproteinase complexed with its endogenous inhibitor pENW

Functional Information from GO Data
ChainGOidnamespacecontents
A0004222molecular_functionmetalloendopeptidase activity
A0006508biological_processproteolysis
A0008237molecular_functionmetallopeptidase activity
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD A 981
ChainResidue
AHIS144
AHIS148
AHIS154
BTRP253
BHOH413

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD A 982
ChainResidue
AHOH349
AHIS36
AASP156
AASP158
AHOH348

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD A 983
ChainResidue
AASP181
AASP185
AHOH325
AHOH431
AHOH433

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD A 984
ChainResidue
AHIS18
AHOH583
AHOH721
AHOH821

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 985
ChainResidue
AGLN7
AASN50
AHOH319
AHOH320
AHOH438
AHOH666

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CD A 986
ChainResidue
AASP194
AHOH442
AHOH571

site_idAC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 987
ChainResidue
APRO203
AHOH392
AHOH598
AHOH746
AHOH747
AHOH837

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD A 988
ChainResidue
AHIS131
AHOH354
AHOH355
AHOH356
AHOH424

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 989
ChainResidue
AHOH380
AHOH386
AHOH550
AHOH551
AHOH552
AHOH836

site_idBC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 990
ChainResidue
AGLU85
AGLU85
AHOH617
AHOH617
AHOH618
AHOH618

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 991
ChainResidue
AGLU85
AGLU85
AGLU121
AHOH455
AHOH803
AHOH803

Functional Information from PROSITE/UniProt
site_idPS00142
Number of Residues10
DetailsZINC_PROTEASE Neutral zinc metallopeptidases, zinc-binding region signature. TMTHELGHNL
ChainResidueDetails
ATHR141-LEU150

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000255|PROSITE-ProRule:PRU00276
ChainResidueDetails
AALA139

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000269|PubMed:12071970, ECO:0007744|PDB:1KUG, ECO:0007744|PDB:1KUK
ChainResidueDetails
ATHR101
ACYS162

site_idSWS_FT_FI3
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12071970, ECO:0000269|PubMed:12077431, ECO:0007744|PDB:1KUF, ECO:0007744|PDB:1KUG, ECO:0007744|PDB:1KUI, ECO:0007744|PDB:1KUK
ChainResidueDetails
AVAL138
AMET142
AHIS148

218853

PDB entries from 2024-04-24

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