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1ILH

Crystal Structure of Human Pregnane X Receptor Ligand Binding Domain Bound to SR12813

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues21
DetailsBINDING SITE FOR RESIDUE SRL A 1
ChainResidue
ALEU206
APHE251
APHE281
ACYS284
AGLN285
APHE288
ATRP299
AMET323
ALEU324
AHIS407
AARG410
ASER208
APHE420
AHOH1595
ALEU209
AVAL211
ALEU240
AMET243
AALA244
AMET246
ASER247

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407

218853

PDB entries from 2024-04-24

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