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1ILH

Crystal Structure of Human Pregnane X Receptor Ligand Binding Domain Bound to SR12813

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues21
DetailsBINDING SITE FOR RESIDUE SRL A 1
ChainResidue
ALEU206
APHE251
APHE281
ACYS284
AGLN285
APHE288
ATRP299
AMET323
ALEU324
AHIS407
AARG410
ASER208
APHE420
AHOH1595
ALEU209
AVAL211
ALEU240
AMET243
AALA244
AMET246
ASER247

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

244693

PDB entries from 2025-11-12

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