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1A52

ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN COMPLEXED TO ESTRADIOL

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EST A 1
ChainResidue
AGLU353
ALEU387
ALEU391
AARG394
AHIS524
ALEU525

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EST B 2
ChainResidue
BLEU391
BARG394
BHIS524
BLEU525
BLEU346
BGLU353
BLEU387

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE AU A 2
ChainResidue
ATYR459
AHIS476
BARG434

site_idAC4
Number of Residues1
DetailsBINDING SITE FOR RESIDUE AU A 3
ChainResidue
ACYS381

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE AU A 5
ChainResidue
APHE337
ACYS417
AHOH562

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE AU B 12
ChainResidue
AARG434
BHIS476

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE AU B 13
ChainResidue
AHIS516
BCYS381

site_idAC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE AU B 15
ChainResidue
BHOH39
BHOH40
BCYS417

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
BTYR537

site_idSWS_FT_FI2
Number of Residues2
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447

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PDB entries from 2024-05-01

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