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5U69

Polycomb protein EED in complex with inhibitor: (3R,4S)-1-[(2-methoxyphenyl)methyl]-N,N-dimethyl-4-(1-methylindol-3-yl)pyrrolidin-3-amine

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsCLSI BEAMLINE 08ID-1
Synchrotron siteCLSI
Beamline08ID-1
Temperature [K]100
Detector technologyCCD
Collection date2013-05-19
DetectorRAYONIX MX-300
Wavelength(s)0.9795
Spacegroup nameP 21 21 21
格子定数 [Å]58.047, 85.400, 91.977
格子定数 [度]90.00, 90.00, 90.00
精密化法
残基62.580 - 1.280
R因子0.13405
Rwork0.133
R-free0.15211
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)5k0m
結合長の平均二乗偏差(RMSD) [Å]0.007
結合角の平均二乗偏差(RMSD) [度]1.424
Data reduction softwareHKL-2000
Data scaling softwareHKL-2000
Phasing softwarePHASER
Refinement softwareREFMAC (5.8.0158)
Quality characteristics
 OverallOuter shell
分解能 [Å] (低)62.5801.330
分解能 [Å] (高)1.2801.280
Rmerge_l_obs0.0770.756
独立反射数118159
<I/σ(I)>9.82.9
完全性 [%]99.899.7
冗長性5.95.7
結晶化条件
結晶ID方法pH温度溶液条件
1VAPOR DIFFUSION8.52903.08M Sodium Formate, 20% Glycerol, 0.1M Tris pH8.5

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件を2024-09-18に公開中

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