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4XP9

X-ray structure of Drosophila dopamine transporter bound to psychostimulant D-amphetamine

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsALS BEAMLINE 8.2.1
Synchrotron siteALS
Beamline8.2.1
Temperature [K]100
Detector technologyCCD
Collection date2014-09-19
DetectorADSC QUANTUM 315r
Wavelength(s)1.00
Spacegroup nameP 21 21 21
Unit cell lengths97.348, 140.748, 166.760
Unit cell angles90.00, 90.00, 90.00
Refinement procedure
Resolution46.720 - 2.800
R-factor0.212
Rwork0.211
R-free0.24200
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)4m48
RMSD bond length0.007
RMSD bond angle1.168
Data reduction softwareXDS
Data scaling softwareXSCALE
Phasing softwarePHASER
Refinement softwarePHENIX
Data quality characteristics
 Overall
Low resolution limit [Å]50.000
High resolution limit [Å]2.800
Number of reflections55464
<I/σ(I)>18.1
Completeness [%]96.6
Redundancy3.7
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, HANGING DROP7277PEG 600 (36%), MOPS (0.1M)

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