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4FA2

Human P38 alpha Mitogen-Activated Kinase In Complex With SB239063

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsAPS BEAMLINE 21-ID-F
Synchrotron siteAPS
Beamline21-ID-F
Temperature [K]100
Detector technologyCCD
Collection date2011-11-09
DetectorMARMOSAIC 225 mm CCD
Wavelength(s)0.97872
Spacegroup nameP 21 21 21
Unit cell lengths65.113, 74.133, 77.770
Unit cell angles90.00, 90.00, 90.00
Refinement procedure
Resolution29.810 - 2.000
R-factor0.17423
Rwork0.172
R-free0.21454
Structure solution methodMOLECULAR REPLACEMENT
RMSD bond length0.012
RMSD bond angle1.332
Data reduction softwareHKL-2000
Data scaling softwareHKL-2000
Phasing softwarePHASER
Refinement softwareREFMAC (5.5.0102)
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]30.0002.030
High resolution limit [Å]2.0002.000
Rmerge0.0590.440
Number of reflections26070
<I/σ(I)>4.87
Completeness [%]99.9100
Redundancy7.37.4
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, SITTING DROP5.52950.1M Ammonium Acetate, 0.1 M BIS-TRIS pH 5.5, 17% PEG 10000, VAPOR DIFFUSION, SITTING DROP, temperature 295K

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