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4B7P

Structure of HSP90 with NMS-E973 inhibitor bound

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsESRF BEAMLINE ID23-2
Synchrotron siteESRF
BeamlineID23-2
Temperature [K]100
Detector technologyCCD
Collection date2009-02-12
DetectorMARMOSAIC 225 mm CCD
Spacegroup nameP 1 21 1
格子定数 [Å]52.746, 44.042, 53.621
格子定数 [度]90.00, 115.59, 90.00
精密化法
残基30.340 - 1.700
R因子0.17549
Rwork0.174
R-free0.19720
Structure solution methodMOLECULAR REPLACEMENT
結合長の平均二乗偏差(RMSD) [Å]0.014
結合角の平均二乗偏差(RMSD) [度]1.866
Data reduction softwareDENZO
Data scaling softwareSCALEPACK
Refinement softwareREFMAC (5.6.0117)
Quality characteristics
 OverallOuter shell
分解能 [Å] (低)30.0001.800
分解能 [Å] (高)1.7001.700
Rmerge_l_obs0.0400.200
独立反射数24199
<I/σ(I)>17
完全性 [%]98.396.9
冗長性4
結晶化条件
結晶ID方法pH温度溶液条件
1

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件を2024-09-18に公開中

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