1HBV
A CHECK ON RATIONAL DRUG DESIGN. CRYSTAL STRUCTURE OF A COMPLEX OF HIV-1 PROTEASE WITH A NOVEL GAMMA-TURN MIMETIC
Experimental procedure
Detector technology | AREA DETECTOR |
Collection date | 1993-12-08 |
Detector | SIEMENS |
Spacegroup name | P 61 |
Unit cell lengths | 63.400, 63.400, 83.900 |
Unit cell angles | 90.00, 90.00, 120.00 |
Refinement procedure
Resolution | 10.000 - 2.300 |
R-factor | 0.177 |
RMSD bond length | 0.018 |
RMSD bond angle | 3.550 |
Data reduction software | XENGEN |
Phasing software | X-PLOR |
Refinement software | PROLSQ |
Data quality characteristics
Overall | |
Low resolution limit [Å] | 9999.000 * |
High resolution limit [Å] | 2.300 * |
Rmerge | 0.095 |
Total number of observations | 36970 * |
Number of reflections | 8051 |
Completeness [%] | 94.0 |
Crystallization Conditions
crystal ID | method | pH | temperature | details |
1 | Vapor diffusion, hanging drop * |
Crystallization Reagents in Literatures
ID | crystal ID | solution | reagent name | concentration (unit) | details |
1 | 1 | reservoir | ammonium sulfate | 16-28 (%) | precipitant |
2 | 1 | reservoir | sodium acetate | 200 (mM) | precipitant |