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1FVV

THE STRUCTURE OF CDK2/CYCLIN A IN COMPLEX WITH AN OXINDOLE INHIBITOR

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsAPS BEAMLINE 17-ID
Synchrotron siteAPS
Beamline17-ID
Temperature [K]100
Detector technologyCCD
Collection date2000-01-03
DetectorMARRESEARCH
Spacegroup nameP 62 2 2
格子定数 [Å]184.952, 184.952, 212.832
格子定数 [度]90.00, 90.00, 120.00
精密化法
残基20.000 - 2.800
R因子0.21
Rwork0.260
R-free0.26000
結合長の平均二乗偏差(RMSD) [Å]0.009

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結合角の平均二乗偏差(RMSD) [度]1.390

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Data scaling softwareHKL-2000
Phasing softwareCNS
Refinement softwareCNS
Quality characteristics
 OverallOuter shell
分解能 [Å] (低)20.0002.980
分解能 [Å] (高)2.8002.800
Rmerge_l_obs0.0700.290
Total number of observations541713

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独立反射数50936
<I/σ(I)>36
完全性 [%]95.990.2
冗長性109
結晶化条件
結晶ID方法pH温度溶液条件
1VAPOR DIFFUSION, HANGING DROP7.5

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20

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Shewchuk L., (2000) J. Med. Chem., 43, 133.

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文献の結晶化試薬
ID結晶ID溶液試薬名濃度 (単位) (単位)詳細
11dropprotein10 (mg/ml)
21dropHEPES20 (mM)
31dropEDTA1 (mM)
41reservoirPEG334010 (%)

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件を2024-09-18に公開中

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