登録情報 | データベース: PDB / ID: 6knr |
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タイトル | Crystal structure of Estrogen-related receptor gamma ligand-binding domain with DN200699 |
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要素 | Estrogen-related receptor gamma |
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キーワード | TRANSCRIPTION / Estrogen-related receptor gamma |
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機能・相同性 | 機能・相同性情報
AF-2 domain binding / nuclear steroid receptor activity / retinoic acid receptor signaling pathway / estrogen response element binding / nuclear receptor-mediated steroid hormone signaling pathway / steroid binding / Nuclear Receptor transcription pathway / nuclear receptor activity / sequence-specific double-stranded DNA binding / positive regulation of cold-induced thermogenesis ...AF-2 domain binding / nuclear steroid receptor activity / retinoic acid receptor signaling pathway / estrogen response element binding / nuclear receptor-mediated steroid hormone signaling pathway / steroid binding / Nuclear Receptor transcription pathway / nuclear receptor activity / sequence-specific double-stranded DNA binding / positive regulation of cold-induced thermogenesis / DNA-binding transcription activator activity, RNA polymerase II-specific / DNA-binding transcription factor activity, RNA polymerase II-specific / regulation of DNA-templated transcription / chromatin / regulation of transcription by RNA polymerase II / positive regulation of transcription by RNA polymerase II / zinc ion binding / nucleoplasm / identical protein binding類似検索 - 分子機能 Oestrogen-related receptor / Retinoic acid receptor / Estrogen receptor/oestrogen-related receptor / Nuclear hormone receptor / Nuclear hormones receptors DNA-binding region signature. / Zinc finger, nuclear hormone receptor-type / Zinc finger, C4 type (two domains) / Nuclear hormone receptors DNA-binding domain profile. / c4 zinc finger in nuclear hormone receptors / Nuclear hormone receptor, ligand-binding domain ...Oestrogen-related receptor / Retinoic acid receptor / Estrogen receptor/oestrogen-related receptor / Nuclear hormone receptor / Nuclear hormones receptors DNA-binding region signature. / Zinc finger, nuclear hormone receptor-type / Zinc finger, C4 type (two domains) / Nuclear hormone receptors DNA-binding domain profile. / c4 zinc finger in nuclear hormone receptors / Nuclear hormone receptor, ligand-binding domain / Nuclear hormone receptor-like domain superfamily / Ligand-binding domain of nuclear hormone receptor / Nuclear receptor (NR) ligand-binding (LBD) domain profile. / Ligand binding domain of hormone receptors / Zinc finger, NHR/GATA-type類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 2.804 Å |
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データ登録者 | Yoon, H. / Kim, J. / Chin, J. / Song, J. / Cho, S.J. |
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引用 | ジャーナル: Eur.J.Med.Chem. / 年: 2020 タイトル: An orally available inverse agonist of estrogen-related receptor gamma showed expanded efficacy for the radioiodine therapy of poorly differentiated thyroid cancer. 著者: Kim, J. / Hwang, H. / Yoon, H. / Lee, J.E. / Oh, J.M. / An, H. / Ji, H.D. / Lee, S. / Cha, E. / Ma, M.J. / Kim, D.S. / Lee, S.J. / Kadayat, T.M. / Song, J. / Lee, S.W. / Jeon, J.H. / Park, K. ...著者: Kim, J. / Hwang, H. / Yoon, H. / Lee, J.E. / Oh, J.M. / An, H. / Ji, H.D. / Lee, S. / Cha, E. / Ma, M.J. / Kim, D.S. / Lee, S.J. / Kadayat, T.M. / Song, J. / Lee, S.W. / Jeon, J.H. / Park, K.G. / Lee, I.K. / Jeon, Y.H. / Chin, J. / Cho, S.J. |
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履歴 | 登録 | 2019年8月7日 | 登録サイト: PDBJ / 処理サイト: PDBJ |
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改定 1.0 | 2020年8月12日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2020年8月19日 | Group: Database references / カテゴリ: citation Item: _citation.page_first / _citation.page_last ..._citation.page_first / _citation.page_last / _citation.pdbx_database_id_PubMed / _citation.title |
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改定 1.2 | 2023年11月22日 | Group: Data collection / Database references / Refinement description カテゴリ: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession |
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