Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
1VTR
DownloadVisualize
BU of 1vtr by Molmil
STRUCTURE OF THE DEOXYTETRANUCLEOTIDE D-PAPTPAPT AND A SEQUENCE-DEPENDENT MODEL FOR POLY(DA-DT)
Descriptor: DNA (5'-D(*AP*TP*AP*T)-3')
Authors:Viswamitra, M.A, Shakked, Z, Jones, P.G, Sheldrick, G.M, Salisbury, S.A, Kennard, O.
Deposit date:1988-08-18
Release date:2011-07-13
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.04 Å)
Cite:Structure of the Deoxytetranucleotide d-pApTpApT and a Sequence-Dependent Model for Poly(dA-dT)
Biopolymers, 21, 1982
1EZT
DownloadVisualize
BU of 1ezt by Molmil
HIGH-RESOLUTION SOLUTION STRUCTURE OF FREE RGS4 BY NMR
Descriptor: REGULATOR OF G-PROTEIN SIGNALING 4
Authors:Moy, F.J, Chanda, P.K, Cockett, M.I, Edris, W, Jones, P.G, Mason, K, Semus, S, Powers, R.
Deposit date:2000-05-11
Release date:2001-01-15
Last modified:2024-05-22
Method:SOLUTION NMR
Cite:NMR structure of free RGS4 reveals an induced conformational change upon binding Galpha.
Biochemistry, 39, 2000
1EZY
DownloadVisualize
BU of 1ezy by Molmil
HIGH-RESOLUTION SOLUTION STRUCTURE OF FREE RGS4 BY NMR
Descriptor: REGULATOR OF G-PROTEIN SIGNALING 4
Authors:Moy, F.J, Chanda, P.K, Cockett, M.I, Edris, W, Jones, P.G, Mason, K, Semus, S, Powers, R.
Deposit date:2000-05-12
Release date:2001-01-15
Last modified:2024-05-22
Method:SOLUTION NMR
Cite:NMR structure of free RGS4 reveals an induced conformational change upon binding Galpha.
Biochemistry, 39, 2000
4YLJ
DownloadVisualize
BU of 4ylj by Molmil
Crystal structure of DYRK1A in complex with 10-Iodo-substituted 11H-indolo[3,2-c]quinoline-6-carboxylic acid inhibitor 5j
Descriptor: 10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, SULFATE ION, ...
Authors:Chaikuad, A, Falke, H, Nowak, R, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2015-03-05
Release date:2015-03-25
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.58 Å)
Cite:10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A.
J.Med.Chem., 58, 2015
4YQH
DownloadVisualize
BU of 4yqh by Molmil
2-[2-(4-Phenyl-1H-imidazol-2-yl)ethyl]quinoxaline (Sunovion Compound 14) co-crystallized with PDE10A
Descriptor: 2-[2-(4-phenyl-1H-imidazol-2-yl)ethyl]quinoxaline, MAGNESIUM ION, ZINC ION, ...
Authors:Burdi, D, Herman, L, Wang, T.
Deposit date:2015-03-13
Release date:2015-04-29
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.308 Å)
Cite:Evolution and synthesis of novel orally bioavailable inhibitors of PDE10A.
Bioorg.Med.Chem.Lett., 25, 2015
4YS7
DownloadVisualize
BU of 4ys7 by Molmil
Co-crystal structure of 2-[2-(5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl]-3-methyl-3H-imidazo[4,5-f]quinoline (compound 39) with PDE10A
Descriptor: 2-[2-(5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl)ethyl]-3-methyl-3H-imidazo[4,5-f]quinoline, MAGNESIUM ION, ZINC ION, ...
Authors:Burdi, D.F, Herman, L, Wang, T.
Deposit date:2015-03-16
Release date:2015-04-29
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.502 Å)
Cite:Evolution and synthesis of novel orally bioavailable inhibitors of PDE10A.
Bioorg.Med.Chem.Lett., 25, 2015
4YLL
DownloadVisualize
BU of 4yll by Molmil
Crystal structure of DYRK1AA in complex with 10-Bromo-substituted 11H-indolo[3,2-c]quinolone-6-carboxylic acid inhibitor 5t
Descriptor: 1,2-ETHANEDIOL, 10-bromo-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ...
Authors:Chaikuad, A, Falke, H, Krojer, T, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2015-03-05
Release date:2015-03-25
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A.
J.Med.Chem., 58, 2015
4YLK
DownloadVisualize
BU of 4ylk by Molmil
Crystal structure of DYRK1A in complex with 10-Chloro-substituted 11H-indolo[3,2-c]quinolone-6-carboxylic acid inhibitor 5s
Descriptor: 1,2-ETHANEDIOL, 10-chloro-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ...
Authors:Chaikuad, A, Falke, H, Krojer, T, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2015-03-05
Release date:2015-03-25
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A.
J.Med.Chem., 58, 2015

225158

PDB entries from 2024-09-18

PDB statisticsPDBj update infoContact PDBjnumon