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5VB2
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BU of 5vb2 by Molmil
Crystal structure of the NavAb voltage-gated sodium channel in a closed conformation
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, CHLORIDE ION, ...
著者Lenaeus, M.J, Catterall, W.A.
登録日2017-03-28
公開日2017-04-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structures of closed and open states of a voltage-gated sodium channel.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
4F4L
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BU of 4f4l by Molmil
Open Channel Conformation of a Voltage Gated Sodium Channel
分子名称: Ion transport protein
著者McCusker, E.C, Bagneris, C, Naylor, C.E, Cole, A.R, D'Avanzo, N, Nichols, C.G, Wallace, B.A.
登録日2012-05-10
公開日2012-10-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.49 Å)
主引用文献Structure of a bacterial voltage-gated sodium channel pore reveals mechanisms of opening and closing.
Nat Commun, 3, 2012
5OQK
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BU of 5oqk by Molmil
Solution NMR structure of truncated, human Hv1/VSOP (Voltage-gated proton channel)
分子名称: Voltage-gated hydrogen channel 1
著者Bayrhuber, M, Maslennikov, I, Kwiatowski, W, Sobol, A, Wierschem, C, Eichmann, C, Riek, R.
登録日2017-08-12
公開日2019-04-03
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Nuclear Magnetic Resonance Solution Structure and Functional Behavior of the Human Proton Channel.
Biochemistry, 58, 2019
2A0L
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BU of 2a0l by Molmil
Crystal structure of KvAP-33H1 Fv complex
分子名称: 33H1 Fv fragment, POTASSIUM ION, Voltage-gated potassium channel
著者Lee, S.Y, Lee, A, Chen, J, Mackinnon, R.
登録日2005-06-16
公開日2005-11-01
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3.9 Å)
主引用文献Structure of the KvAP voltage-dependent K+ channel and its dependence on the lipid membrane.
Proc.Natl.Acad.Sci.Usa, 102, 2005
2KYH
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BU of 2kyh by Molmil
Solution structure of the voltage-sensing domain of KvAP
分子名称: Voltage-gated potassium channel
著者Butterwick, J.A, MacKinnon, R.
登録日2010-05-26
公開日2010-09-29
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Solution Structure and Phospholipid Interactions of the Isolated Voltage-Sensor Domain from KvAP.
J.Mol.Biol., 403, 2010
5KMF
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BU of 5kmf by Molmil
Structure of CavAb in complex with nimodipine
分子名称: 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-26
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
5KLG
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BU of 5klg by Molmil
Structure of CavAb(W195Y) in complex with Br-dihydropyridine derivative UK-59811
分子名称: 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-24
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
3ZJZ
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BU of 3zjz by Molmil
Open-form NavMS Sodium Channel Pore (with C-terminal Domain)
分子名称: DODECAETHYLENE GLYCOL, HEGA-10, ION TRANSPORT PROTEIN, ...
著者Bagneris, C, Naylor, C.E, Wallace, B.A.
登録日2013-01-21
公開日2013-10-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.92 Å)
主引用文献Role of the C-Terminal Domain in the Structure and Function of Tetrameric Sodium Channels.
Nat.Commun., 4, 2013
5BZB
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BU of 5bzb by Molmil
NavMs voltage-gated sodium channel pore and C-terminal domain
分子名称: DODECAETHYLENE GLYCOL, HEGA-10, Ion transport protein, ...
著者Naylor, C.E, Bagneris, C, Wallace, B.A.
登録日2015-06-11
公開日2016-02-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Molecular basis of ion permeability in a voltage-gated sodium channel.
Embo J., 35, 2016
4X8A
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BU of 4x8a by Molmil
NavMS pore and C-terminal domain grown from protein purified in LiCl
分子名称: HEGA-10, Ion transport protein, NONAETHYLENE GLYCOL, ...
著者Naylor, C.E, Bagneris, C, Wallace, B.A.
登録日2014-12-10
公開日2016-03-09
最終更新日2017-08-30
実験手法X-RAY DIFFRACTION (3.02 Å)
主引用文献Molecular basis of ion permeability in a voltage-gated sodium channel.
Embo J., 35, 2016
4X88
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BU of 4x88 by Molmil
E178D Selectivity filter mutant of NavMS voltage-gated pore
分子名称: HEGA-10, Ion transport protein, PENTAETHYLENE GLYCOL, ...
著者Naylor, C.E, Bagneris, C, Wallace, B.A.
登録日2014-12-10
公開日2016-02-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Molecular basis of ion permeability in a voltage-gated sodium channel.
Embo J., 35, 2016
4X89
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BU of 4x89 by Molmil
NavMs voltage-gated sodium channal pore and C-terminal domain soaked with Silver nitrate
分子名称: HEGA-10, Ion transport protein, PENTAETHYLENE GLYCOL, ...
著者Naylor, C.E, Bagneris, C, Wallace, B.A.
登録日2014-12-10
公開日2016-03-09
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Molecular basis of ion permeability in a voltage-gated sodium channel.
Embo J., 35, 2016
3RVZ
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BU of 3rvz by Molmil
Crystal structure of the NavAb voltage-gated sodium channel (Ile217Cys, 2.8 A)
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Ion transport protein
著者Payandeh, J, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2011-05-06
公開日2011-07-13
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The crystal structure of a voltage-gated sodium channel.
Nature, 475, 2011
3RW0
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BU of 3rw0 by Molmil
Crystal structure of the NavAb voltage-gated sodium channel (Met221Cys, 2.95 A)
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Ion transport protein
著者Payandeh, J, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2011-05-06
公開日2011-07-13
最終更新日2011-07-27
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献The crystal structure of a voltage-gated sodium channel.
Nature, 475, 2011
3RVY
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BU of 3rvy by Molmil
Crystal structure of the NavAb voltage-gated sodium channel (Ile217Cys, 2.7 A)
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Ion transport protein
著者Payandeh, J, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2011-05-06
公開日2011-07-13
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The crystal structure of a voltage-gated sodium channel.
Nature, 475, 2011
4G7Y
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BU of 4g7y by Molmil
Crystal structure of voltage sensing domain of Ci-VSP with fragment antibody (R217E, 2.8 A)
分子名称: CHLORIDE ION, Fragment antibody heavy chain, Fragment antibody light chain, ...
著者Li, Q.
登録日2012-07-20
公開日2014-02-05
最終更新日2019-07-17
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural mechanism of voltage-dependent gating in an isolated voltage-sensing domain.
Nat. Struct. Mol. Biol., 21, 2014
5KMD
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BU of 5kmd by Molmil
Structure of CavAb in complex with amlodipine
分子名称: 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-26
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
5KLB
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BU of 5klb by Molmil
Crystal structure of the CavAb voltage-gated calcium channel(wild-type, 2.7A)
分子名称: 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, CALCIUM ION, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-23
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
5KLS
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BU of 5kls by Molmil
Structure of CavAb in complex with Br-dihydropyridine derivative UK-59811
分子名称: 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-25
公開日2016-08-31
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.299 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
5KMH
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BU of 5kmh by Molmil
Structure of CavAb in complex with Br-verapamil
分子名称: (2~{R})-2-(2-bromophenyl)-5-[2-(3,4-dimethoxyphenyl)ethyl-methyl-amino]-2-propan-2-yl-pentanenitrile, 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIPALMITOYL-SN-GLYCERO-3-PHOSPHATE, ...
著者Tang, L, Gamal EL-Din, T.M, Swanson, T.M, Pryde, D.C, Scheuer, T, Zheng, N, Catterall, W.A.
登録日2016-06-27
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural basis for inhibition of a voltage-gated Ca(2+) channel by Ca(2+) antagonist drugs.
Nature, 537, 2016
4G80
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BU of 4g80 by Molmil
Crystal structure of voltage sensing domain of Ci-VSP with fragment antibody (WT, 3.8 A)
分子名称: Voltage-sensor containing phosphatase, fragment antibody heavy chain, fragment antibody light chain
著者Li, Q.
登録日2012-07-20
公開日2014-02-05
最終更新日2017-12-13
実験手法X-RAY DIFFRACTION (3.58 Å)
主引用文献Structural mechanism of voltage-dependent gating in an isolated voltage-sensing domain.
Nat. Struct. Mol. Biol., 21, 2014
4G7V
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BU of 4g7v by Molmil
Crystal structure of voltage sensing domain of Ci-VSP with fragment antibody (R217E, 2.5 A)
分子名称: CHLORIDE ION, LAURYL DIMETHYLAMINE-N-OXIDE, SUCCINIC ACID, ...
著者Li, Q.
登録日2012-07-20
公開日2014-02-05
最終更新日2017-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural mechanism of voltage-dependent gating in an isolated voltage-sensing domain.
Nat. Struct. Mol. Biol., 21, 2014
4BGN
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BU of 4bgn by Molmil
cryo-EM structure of the NavCt voltage-gated sodium channel
分子名称: VOLTAGE-GATED SODIUM CHANNEL
著者Tsai, C.J, Tani, K, Irie, K, Hiroaki, Y, Shimomura, T, Mcmillan, D.G, Cook, G.M, Schertler, G, Fujiyoshi, Y, Li, X.D.
登録日2013-03-28
公開日2013-07-10
最終更新日2023-12-20
実験手法ELECTRON CRYSTALLOGRAPHY (9 Å)
主引用文献Two Alternative Conformations of a Voltage-Gated Sodium Channel.
J.Mol.Biol., 425, 2013
4DXW
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BU of 4dxw by Molmil
Crystal structure of NavRh, a voltage-gated sodium channel
分子名称: 1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, Ion transport protein, ...
著者Zhang, X, Ren, W.L, Yan, C.Y, Wang, J.W, Yan, N.
登録日2012-02-28
公開日2012-05-23
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3.052 Å)
主引用文献Crystal structure of an orthologue of the NaChBac voltage-gated sodium channel
Nature, 486, 2012
4CBC
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BU of 4cbc by Molmil
Open-form NavMS Sodium Channel Pore (with C-terminal Domain) after thallium soak
分子名称: HEGA-10, ION TRANSPORT PROTEIN, SODIUM ION
著者Bagneris, C, Naylor, C.E, Wallace, B.A.
登録日2013-10-12
公開日2014-05-28
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.664 Å)
主引用文献Prokaryotic Navms Channel as a Structural and Functional Model for Eukaryotic Sodium Channel Antagonism.
Proc.Natl.Acad.Sci.USA, 111, 2014

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