8AX3
Structure of recombinant human beta-glucocerebrosidase in complex with L-carbaxylosyl fluoride
Summary for 8AX3
Entry DOI | 10.2210/pdb8ax3/pdb |
Related | 8AWK 8AWR |
Descriptor | Lysosomal acid glucosylceramidase, CALCIUM ION, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (11 entities in total) |
Functional Keywords | beta-glucocerebrosidase, glycoside hydrolase, inhibitor, carbasugar, pharmacological chaperone, hydrolase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 117599.60 |
Authors | |
Primary citation | Bhosale, S.,Kandalkar, S.,Gilormini, P.A.,Akintola, O.,Rowland, R.J.,Adabala, P.J.P.,King, D.,Deen, M.C.,Xi, K.,Davies, G.J.,Vocadlo, D.J.,Bennet, A.J. Single turnover covalent inhibitors for functional chaperoning of lysosomal glycoside hydrolases To be published, |
Experimental method | X-RAY DIFFRACTION (1.59 Å) |
Structure validation
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