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8A66

Crystal structure of MST2 in complex with XMU-MP-1

Summary for 8A66
Entry DOI10.2210/pdb8a66/pdb
DescriptorSerine/threonine-protein kinase 3 36kDa subunit, 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5H-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide, SODIUM ION, ... (5 entities in total)
Functional Keywordsserine/threonine kinase, autophosrylation, transferase, transcription
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight68886.63
Authors
Nawrotek, A.,Vuillard, L.,Miallau, L.,Weber, C. (deposition date: 2022-06-16, release date: 2022-07-20, Last modification date: 2022-12-07)
Primary citationWeber, C.,Vuillard, L.,Delerive, P.,Miallau, L.,Nawrotek, A.
Crystal structure of the Kelch domain of human Keap1in complex with ligand S217879
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.901 Å)
Structure validation

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