5J5X
Complex of PKA with the bisubstrate protein kinase inhibitor ARC-1416
Summary for 5J5X
Entry DOI | 10.2210/pdb5j5x/pdb |
Related | 5IZF 5IZJ |
Descriptor | cAMP-dependent protein kinase catalytic subunit alpha, 47P-AZ1-DAL-DAR-DAR-DAR-DAR, SULFATE ION, ... (5 entities in total) |
Functional Keywords | protein kinase, inhibitor, bisubstrate, oligoarginine, pka, transferase |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 42357.33 |
Authors | Alam, K.A.,Ivan, T.,Uri, A.,Engh, R.A. (deposition date: 2016-04-04, release date: 2016-07-20, Last modification date: 2019-06-19) |
Primary citation | Ivan, T.,Enkvist, E.,Viira, B.,Manoharan, G.B.,Raidaru, G.,Pflug, A.,Alam, K.A.,Zaccolo, M.,Engh, R.A.,Uri, A. Bifunctional Ligands for Inhibition of Tight-Binding Protein-Protein Interactions. Bioconjug.Chem., 27:1900-1910, 2016 Cited by PubMed: 27389935DOI: 10.1021/acs.bioconjchem.6b00293 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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