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5BW2

X-ray crystal structure of Aplysia californica acetylcholine binding protein (Ac-AChBP) Y55W in complex with 2-Pyridin-3-yl-1-aza-bicyclo[2.2.2]octane; 2-(3-pyridyl)quinuclidine; 2-PQ (TI-4699)

Summary for 5BW2
Entry DOI10.2210/pdb5bw2/pdb
Related5BRX
DescriptorSoluble acetylcholine receptor, (2R)-2-(pyridin-3-yl)-1-azabicyclo[2.2.2]octane (3 entities in total)
Functional Keywordsachbp, nicotine, acetylcholine, acetylcholine binding protein
Biological sourceAplysia californica (California sea hare)
Total number of polymer chains5
Total formula weight131928.78
Authors
Bobango, J.,Sankaran, B.,Park, J.F.,Wu, J.,Talley, T.T. (deposition date: 2015-06-05, release date: 2015-06-24, Last modification date: 2023-09-27)
Primary citationBobango, J.,Sankaran, B.,Park, J.F.,Wu, J.,Talley, T.T.
Comparisons of Binding Affinities for Neuronal Nicotinic Receptors (NNRs) and AChBPs
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.27 Å)
Structure validation

220113

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