4LQ3
Crystal structure of human norovirus RNA-dependent RNA-polymerase bound to the inhibitor PPNDS
Summary for 4LQ3
Entry DOI | 10.2210/pdb4lq3/pdb |
Related | 4LQ9 |
Descriptor | RNA-dependent RNA-polymerase, 5'-R(P*GP*G)-3', 3-[(E)-{4-formyl-5-hydroxy-6-methyl-3-[(phosphonooxy)methyl]pyridin-2-yl}diazenyl]-7-nitronaphthalene-1,5-disulfonic acid, ... (5 entities in total) |
Functional Keywords | rna-dependent-rna-polymerase, rdrp-inhibotir complex, viral protein-replication inhibitor-rna complex, viral protein/replication inhibitor/rna |
Biological source | Norovirus |
Total number of polymer chains | 2 |
Total formula weight | 61753.26 |
Authors | Milani, M.,Tarantino, D.,Mastrangelo, E.,Croci, R. (deposition date: 2013-07-17, release date: 2014-02-12, Last modification date: 2024-02-28) |
Primary citation | Tarantino, D.,Pezzullo, M.,Mastrangelo, E.,Croci, R.,Rohayem, J.,Robel, I.,Bolognesi, M.,Milani, M. Naphthalene-sulfonate inhibitors of human norovirus RNA-dependent RNA-polymerase. Antiviral Res., 102:23-28, 2014 Cited by PubMed: 24316032DOI: 10.1016/j.antiviral.2013.11.016 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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