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4EBP

BlaC E166A Cefotaxime Acyl-Intermediate Complex

Summary for 4EBP
Entry DOI10.2210/pdb4ebp/pdb
Related3VFF 3VFH 4EBI 4EBL 4EBM 4EBN 4EBO
DescriptorBeta-lactamase, PHOSPHATE ION, CEFOTAXIME, C3' cleaved, open, bound form, ... (4 entities in total)
Functional Keywordsambler class a beta-lactamase, beta-lactamase, serine hydrolase, esterase, hydrolase-antibiotic complex, structural genomics, tb structural genomics consortium, tbsgc, hydrolase/antibiotic
Biological sourceMycobacterium tuberculosis
Total number of polymer chains4
Total formula weight114508.35
Authors
Mire, J.A.,TB Structural Genomics Consortium (TBSGC) (deposition date: 2012-03-23, release date: 2013-04-03, Last modification date: 2023-09-13)
Primary citationMire, J.A.,Pai, P.,Siddiqi, N.,Russell, D.H.,Rubin, E.J.,Sacchettini, J.C.
Faropenem is Effective Against Mycobacterium tuberculosis in vitro and in vivo
To be Published,
Experimental method
X-RAY DIFFRACTION (2.29 Å)
Structure validation

220113

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