4DVX
Crystal structure of clade A/E 93TH057 HIV-1 gp120 core in complex with MAE-II-188
Summary for 4DVX
Entry DOI | 10.2210/pdb4dvx/pdb |
Related | 4DVR 4DVS 4DVT 4DVU 4DVV 4DVW |
Descriptor | clade A/E 93TH057 HIV-1 gp120 core, 2-acetamido-2-deoxy-beta-D-glucopyranose, N-(4-chloro-3-fluorophenyl)-N'-{[(3R)-1-cyclopropylpyrrolidin-3-yl]methyl}ethanediamide, ... (5 entities in total) |
Functional Keywords | hiv-1 gp120, small molecule inhibitor, cd4 binding site, mae-ii-188, viral protein-transcription inhibitor complex, viral protein/transcription inhibitor |
Biological source | Human immunodeficiency virus 1 |
Total number of polymer chains | 2 |
Total formula weight | 84343.50 |
Authors | Kwon, Y.D.,Kwong, P.D. (deposition date: 2012-02-23, release date: 2013-02-27, Last modification date: 2020-07-29) |
Primary citation | Kwon, Y.D.,Lalonde, J.M.,Yang, Y.,Elban, M.A.,Sugawara, A.,Courter, J.R.,Jones, D.M.,Smith, A.B.,Debnath, A.K.,Kwong, P.D. Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site. Plos One, 9:e85940-e85940, 2014 Cited by PubMed: 24489681DOI: 10.1371/journal.pone.0085940 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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