2ZDX
Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4
Summary for 2ZDX
Entry DOI | 10.2210/pdb2zdx/pdb |
Related | 2ZDY |
Descriptor | Pyruvate dehydrogenase kinase isozyme 4, 4-[4-(4-methoxyphenyl)-5-methyl-1H-pyrazol-3-yl]benzene-1,3-diol (3 entities in total) |
Functional Keywords | pdk4, kinase, atp-binding, inhibitor, carbohydrate metabolism, glucose metabolism, mitochondrion, phosphoprotein, transferase, transit peptide |
Biological source | Homo sapiens (Human) |
Cellular location | Mitochondrion matrix: Q16654 |
Total number of polymer chains | 2 |
Total formula weight | 90134.63 |
Authors | Kawamoto, M.,Shiromizu, I.,Kukimoto-niino, M.,Tokmakov, A.,Terada, T.,Shirouzu, M.,Matsusue, T.,Yokoyama, S. (deposition date: 2007-11-30, release date: 2008-12-09, Last modification date: 2023-11-01) |
Primary citation | Kukimoto-Niino, M.,Tokmakov, A.,Terada, T.,Ohbayashi, N.,Fujimoto, T.,Gomi, S.,Shiromizu, I.,Kawamoto, M.,Matsusue, T.,Shirouzu, M.,Yokoyama, S. Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr.,Sect.D, 67:763-773, 2011 Cited by PubMed: 21904029DOI: 10.1107/S090744491102405X PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.54 Å) |
Structure validation
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