2O64
Crystal structure of Pim1 with Quercetagetin
Summary for 2O64
Entry DOI | 10.2210/pdb2o64/pdb |
Related | 2O3P 2O63 2O65 |
Descriptor | Proto-oncogene serine/threonine-protein kinase Pim-1, IMIDAZOLE, 3,5,6,7-TETRAHYDROXY-2-(3,4-DIHYDROXYPHENYL)-4H-CHROMEN-4-ONE, ... (4 entities in total) |
Functional Keywords | pim1, quercetagetin, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Isoform 2: Cytoplasm. Isoform 1: Cell membrane: P11309 |
Total number of polymer chains | 1 |
Total formula weight | 34288.72 |
Authors | Holder, S.,Zemskova, M.,Zhang, C.,Tabrizizad, M.,Bremer, R.,Neidigh, J.W.,Lilly, M.B. (deposition date: 2006-12-06, release date: 2007-02-13, Last modification date: 2023-12-27) |
Primary citation | Holder, S.,Zemskova, M.,Zhang, C.,Tabrizizad, M.,Bremer, R.,Neidigh, J.W.,Lilly, M.B. Characterization of a potent and selective small-molecule inhibitor of the PIM1 kinase. Mol.Cancer Ther., 6:163-172, 2007 Cited by PubMed: 17218638DOI: 10.1158/1535-7163.MCT-06-0397 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.44 Å) |
Structure validation
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