1HRN
HIGH RESOLUTION CRYSTAL STRUCTURES OF RECOMBINANT HUMAN RENIN IN COMPLEX WITH POLYHYDROXYMONOAMIDE INHIBITORS
1HRN の概要
エントリーDOI | 10.2210/pdb1hrn/pdb |
分子名称 | RENIN, 2-acetamido-2-deoxy-beta-D-glucopyranose, (2R,4S,5S)-N-[(2S,3R,4S)-1-cyclohexyl-3,4-dihydroxy-6-methylheptan-2-yl]-2-(cyclopropylmethyl)-4,5-dihydroxy-6-phenylhexanamide, ... (4 entities in total) |
機能のキーワード | aspartic proteinase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 75329.03 |
構造登録者 | |
主引用文献 | Tong, L.,Pav, S.,Lamarre, D.,Pilote, L.,LaPlante, S.,Anderson, P.C.,Jung, G. High resolution crystal structures of recombinant human renin in complex with polyhydroxymonoamide inhibitors. J.Mol.Biol., 250:211-222, 1995 Cited by PubMed: 7608971DOI: 10.1006/jmbi.1995.0372 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.8 Å) |
構造検証レポート
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