1GAG
CRYSTAL STRUCTURE OF THE INSULIN RECEPTOR KINASE IN COMPLEX WITH A BISUBSTRATE INHIBITOR
Summary for 1GAG
Entry DOI | 10.2210/pdb1gag/pdb |
Related | 1IR3 |
Descriptor | INSULIN RECEPTOR, TYROSINE KINASE DOMAIN, BISUBSTRATE PEPTIDE INHIBITOR, MAGNESIUM ION, ... (5 entities in total) |
Functional Keywords | protein kinase inhibitor, tyrosine kinase, transferase, signaling protein, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Membrane; Single-pass type I membrane protein: P06213 |
Total number of polymer chains | 2 |
Total formula weight | 36985.14 |
Authors | Parang, K.,Till, J.H.,Ablooglu, A.J.,Kohanski, R.A.,Hubbard, S.R.,Cole, P.A. (deposition date: 2000-11-29, release date: 2001-01-17, Last modification date: 2023-11-15) |
Primary citation | Parang, K.,Till, J.H.,Ablooglu, A.J.,Kohanski, R.A.,Hubbard, S.R.,Cole, P.A. Mechanism-based design of a protein kinase inhibitor. Nat.Struct.Biol., 8:37-41, 2001 Cited by PubMed: 11135668DOI: 10.1038/83028 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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