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5J79

The identification and pharmacological characterization of 6-(tert-butylsulfonyl)-N-(5-fluoro-1H-indazol-3-yl)quinolin-4-amine (GSK583), a highly potent and selective inhibitor of RIP2 Kinase, Compound 3 complex

Resources
File formatFile name (file size)
PDBx/mmCIF5j79.cif.gz Display(138.08 KB)
5j79.cif
PDBx/mmJSONall5j79.json.gz Display (Tree)(91.22 KB)
5j79.json
no-atom5j79-noatom.json.gz Display (Header)(17.90 KB)
5j79-noatom.json
add only5j79-plus.json.gz Display(1.47 KB)
5j79-plus.json
PDBMLall5j79.xml.gz Display(184.99 KB)
5j79.xml
no-atom5j79-noatom.xml.gz Display(36.04 KB)
5j79-noatom.xml
ext-atom5j79-extatom.xml.gz Display(112.09 KB)
5j79-extatom.xml
PDBpdb5j79.ent.gz Display(106.36 KB)
pdb5j79.ent
RDF5j79.rdf.gz Visualize(104.40 KB)
5j79.rdf
Structure factorsr5j79sf.ent.gz Display(683.47 KB)
r5j79sf.ent
Biological unit (mmCIF format)5j79-assembly1.cif.gz Display(125.32 KB)
5j79-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)5j79.pdb1.gz Display(100.42 KB)
5j79.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF5j79_validation.pdf.gz Display(1.06 MB)
5j79_validation.pdf
PDF-full5j79_full_validation.pdf.gz Display(1.06 MB)
5j79_full_validation.pdf
mmCIF5j79_validation.cif.gz Display(36.41 KB)
5j79_validation.cif
XML5j79_validation.xml.gz Display(25.26 KB)
5j79_validation.xml
PNG5j79_multipercentile_validation.png.gz Display(164.23 KB)
5j79_multipercentile_validation.png
SVG5j79_multipercentile_validation.svg.gz Display(965.00 B)
5j79_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5j79_validation_2fo-fc_map_coef.cif.gz Display(309.09 KB)
5j79_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5j79_validation_fo-fc_map_coef.cif.gz Display(301.68 KB)
5j79_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5j79_validation_2fo-fc_map_coef.mtz Visualize(735.07 KB)
fo-fc (MTZ)5j79_validation_fo-fc_map_coef.mtz Visualize(735.07 KB)

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PDB entries from 2024-05-15

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