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4UWK

Discovery of (2S)-8-((3R)-3-Methylmorpholin-4-yl)-1-(3-methyl-2-oxo- butyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido(1,2-a)pyrimidin-6- one: a Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors

Resources
File formatFile name (file size)
PDBx/mmCIF4uwk.cif.gz Display(124.94 KB)
4uwk.cif
PDBx/mmJSONall4uwk.json.gz Display (Tree)(84.75 KB)
4uwk.json
no-atom4uwk-noatom.json.gz Display (Header)(15.56 KB)
4uwk-noatom.json
add only4uwk-plus.json.gz Display(967.00 B)
4uwk-plus.json
PDBMLall4uwk.xml.gz Display(166.62 KB)
4uwk.xml
no-atom4uwk-noatom.xml.gz Display(31.90 KB)
4uwk-noatom.xml
ext-atom4uwk-extatom.xml.gz Display(101.61 KB)
4uwk-extatom.xml
PDBpdb4uwk.ent.gz Display(95.31 KB)
pdb4uwk.ent
RDF4uwk.rdf.gz Visualize(100.22 KB)
4uwk.rdf
Structure factorsr4uwksf.ent.gz Display(222.31 KB)
r4uwksf.ent
Biological unit (mmCIF format)4uwk-assembly1.cif.gz Display(116.48 KB)
4uwk-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4uwk.pdb1.gz Display(90.51 KB)
4uwk.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4uwk_validation.pdf.gz Display(860.37 KB)
4uwk_validation.pdf
PDF-full4uwk_full_validation.pdf.gz Display(865.87 KB)
4uwk_full_validation.pdf
mmCIF4uwk_validation.cif.gz Display(28.67 KB)
4uwk_validation.cif
XML4uwk_validation.xml.gz Display(20.68 KB)
4uwk_validation.xml
PNG4uwk_multipercentile_validation.png.gz Display(165.78 KB)
4uwk_multipercentile_validation.png
SVG4uwk_multipercentile_validation.svg.gz Display(971.00 B)
4uwk_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4uwk_validation_2fo-fc_map_coef.cif.gz Display(200.87 KB)
4uwk_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4uwk_validation_fo-fc_map_coef.cif.gz Display(196.45 KB)
4uwk_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4uwk_validation_2fo-fc_map_coef.mtz Visualize(484.41 KB)
fo-fc (MTZ)4uwk_validation_fo-fc_map_coef.mtz Visualize(484.41 KB)

219869

PDB entries from 2024-05-15

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