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3VAP

Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity

Resources
File formatFile name (file size)
PDBx/mmCIF3vap.cif.gz Display(217.14 KB)
3vap.cif
PDBx/mmJSONall3vap.json.gz Display (Tree)(145.46 KB)
3vap.json
no-atom3vap-noatom.json.gz Display (Header)(12.36 KB)
3vap-noatom.json
add only3vap-plus.json.gz Display(1.43 KB)
3vap-plus.json
PDBMLall3vap.xml.gz Display(290.93 KB)
3vap.xml
no-atom3vap-noatom.xml.gz Display(23.32 KB)
3vap-noatom.xml
ext-atom3vap-extatom.xml.gz Display(92.79 KB)
3vap-extatom.xml
PDBpdb3vap.ent.gz Display(177.17 KB)
pdb3vap.ent
RDF3vap.rdf.gz Visualize(70.77 KB)
3vap.rdf
Structure factorsr3vapsf.ent.gz Display(203.81 KB)
r3vapsf.ent
Biological unit (mmCIF format)3vap-assembly1.cif.gz Display(209.74 KB)
3vap-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3vap.pdb1.gz Display(171.72 KB)
3vap.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3vap_validation.pdf.gz Display(672.67 KB)
3vap_validation.pdf
PDF-full3vap_full_validation.pdf.gz Display(675.63 KB)
3vap_full_validation.pdf
mmCIF3vap_validation.cif.gz Display(14.26 KB)
3vap_validation.cif
XML3vap_validation.xml.gz Display(11.27 KB)
3vap_validation.xml
PNG3vap_multipercentile_validation.png.gz Display(167.76 KB)
3vap_multipercentile_validation.png
SVG3vap_multipercentile_validation.svg.gz Display(979.00 B)
3vap_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3vap_validation_2fo-fc_map_coef.cif.gz Display(96.08 KB)
3vap_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3vap_validation_fo-fc_map_coef.cif.gz Display(93.75 KB)
3vap_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3vap_validation_2fo-fc_map_coef.mtz Visualize(235.29 KB)
fo-fc (MTZ)3vap_validation_fo-fc_map_coef.mtz Visualize(235.29 KB)

221051

PDB entries from 2024-06-12

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