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3L17

Discovery of (thienopyrimidin-2-yl)aminopyrimidines as Potent, Selective, and Orally Available Pan-PI3-Kinase and Dual Pan-PI3-Kinase/mTOR Inhibitors for the Treatment of Cancer

Resources
File formatFile name (file size)
PDBx/mmCIF3l17.cif.gz Display(183.10 KB)
3l17.cif
PDBx/mmJSONall3l17.json.gz Display (Tree)(125.96 KB)
3l17.json
no-atom3l17-noatom.json.gz Display (Header)(24.04 KB)
3l17-noatom.json
add only3l17-plus.json.gz Display(1.10 KB)
3l17-plus.json
PDBMLall3l17.xml.gz Display(244.00 KB)
3l17.xml
no-atom3l17-noatom.xml.gz Display(43.70 KB)
3l17-noatom.xml
ext-atom3l17-extatom.xml.gz Display(150.37 KB)
3l17-extatom.xml
PDBpdb3l17.ent.gz Display(140.69 KB)
pdb3l17.ent
RDF3l17.rdf.gz Visualize(133.03 KB)
3l17.rdf
Structure factorsr3l17sf.ent.gz Display(312.61 KB)
r3l17sf.ent
Biological unit (mmCIF format)3l17-assembly1.cif.gz Display(170.98 KB)
3l17-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3l17.pdb1.gz Display(134.14 KB)
3l17.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3l17_validation.pdf.gz Display(734.86 KB)
3l17_validation.pdf
PDF-full3l17_full_validation.pdf.gz Display(762.71 KB)
3l17_full_validation.pdf
mmCIF3l17_validation.cif.gz Display(44.08 KB)
3l17_validation.cif
XML3l17_validation.xml.gz Display(32.51 KB)
3l17_validation.xml
PNG3l17_multipercentile_validation.png.gz Display(167.11 KB)
3l17_multipercentile_validation.png
SVG3l17_multipercentile_validation.svg.gz Display(979.00 B)
3l17_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3l17_validation_2fo-fc_map_coef.cif.gz Display(214.07 KB)
3l17_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3l17_validation_fo-fc_map_coef.cif.gz Display(209.17 KB)
3l17_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3l17_validation_2fo-fc_map_coef.mtz Visualize(493.18 KB)
fo-fc (MTZ)3l17_validation_fo-fc_map_coef.mtz Visualize(493.18 KB)

219140

PDB entries from 2024-05-01

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