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6O5I

Menin in complex with MI-3454

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues21
Detailsbinding site for residue LMY A 601
ChainResidue
ASER155
AASN282
AMET322
ATYR323
ATRP341
AGLU363
AGLU366
AVAL371
ADMS602
AHOH892
AHOH1010
ALEU177
AHOH1129
AHOH1168
ASER178
AHIS181
AALA182
APHE238
ACYS241
ATYR276
AMET278

site_idAC2
Number of Residues3
Detailsbinding site for residue DMS A 602
ChainResidue
ALMY601
AHOH1348
AHOH1428

site_idAC3
Number of Residues6
Detailsbinding site for residue DMS A 603
ChainResidue
AVAL185
AGLY190
AGLU191
ATYR227
AARG229
ASER583

site_idAC4
Number of Residues5
Detailsbinding site for residue DMS A 604
ChainResidue
APHE47
AGLN400
AHOH808
AHOH923
AHOH1014

site_idAC5
Number of Residues5
Detailsbinding site for residue DMS A 605
ChainResidue
ATYR77
AHOH766
AHOH853
AHOH1152
AHOH1531

site_idAC6
Number of Residues4
Detailsbinding site for residue SO4 A 606
ChainResidue
APRO12
AARG14
AHOH744
AHOH790

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 A 607
ChainResidue
ATYR133
APHE134
AARG137
ALYS151

site_idAC8
Number of Residues8
Detailsbinding site for residue SO4 A 608
ChainResidue
AARG332
AVAL334
AARG335
AGLY401
AALA403
AHOH984
AHOH1036
AHOH1134

site_idAC9
Number of Residues7
Detailsbinding site for residue PG4 A 609
ChainResidue
ALEU75
ATHR76
APHE365
AHIS433
AHOH761
AHOH813
AHOH1232

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER543

219869

PDB entries from 2024-05-15

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