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6FS1

MCL1 in complex with an indole acid ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue E4Q A 401
ChainResidue
AMET231
AHOH555
AHOH572
AHOH589
AVAL249
AMET250
AVAL253
AARG263
ATHR266
ALEU267
APHE270
AGLY271

site_idAC2
Number of Residues9
Detailsbinding site for residue EDO B 401
ChainResidue
AARG300
ATHR301
AARG303
AASP304
BARG300
BTHR301
BARG303
BASP304
BHOH588

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO B 402
ChainResidue
BALA204
BALA205
BARG208
BASP313

site_idAC4
Number of Residues12
Detailsbinding site for residue E4Q B 403
ChainResidue
BMET231
BVAL249
BMET250
BVAL253
BARG263
BTHR266
BLEU267
BPHE270
BGLY271
BHOH547
BHOH580
BHOH593

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
BLYS197
ALYS194
ALYS197
BLYS194

219869

PDB entries from 2024-05-15

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