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4A9H

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 1-(2-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one

Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1187
ChainResidue
AGLN94
AHOH2024
BTRP97

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1188
ChainResidue
ATRP97
AASP161
AILE162
AHOH2111
AHOH2131
BGLN94

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE TVP A 1189
ChainResidue
APRO98
ALEU110
AASN156
AILE162
AHOH2061

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE TVP B 1183
ChainResidue
BPRO98
BLEU110
BCYS152
BASN156
BHOH2039

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE TVP C 1183
ChainResidue
CPRO98
CLEU110
CASN156
CILE162
CHOH2032

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 C 1184
ChainResidue
BARG100
CARG128
CASN132
CTYR134

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1190
ChainResidue
AARG100
AHOH2014
AHOH2021

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP112
CTYR155
CASN156
CLYS157
ATYR155
AASN156
ALYS157
BASP112
BTYR155
BASN156
BLYS157
CASP112

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP160
AASP161
BASP160
BASP161
CASP160
CASP161

220113

PDB entries from 2024-05-22

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