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3F9Z

Structural Insights into Lysine Multiple Methylation by SET Domain Methyltransferases, SET8-Y245F / H4-Lys20 / AdoHcy

Functional Information from GO Data
ChainGOidnamespacecontents
A0042799molecular_functionhistone H4K20 methyltransferase activity
B0042799molecular_functionhistone H4K20 methyltransferase activity
C0042799molecular_functionhistone H4K20 methyltransferase activity
D0042799molecular_functionhistone H4K20 methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE SAH A 801
ChainResidue
AHOH87
ALEU296
AASN298
AHIS299
ATYR336
ATRP349
AHOH374
AHOH425
FHIS18
AHOH115
AHOH137
AGLY225
ALYS226
AARG228
ACYS270
ATYR271
AARG295

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE SAH B 801
ChainResidue
BHOH85
BGLY225
BLYS226
BARG228
BCYS270
BTYR271
BLEU296
BASN298
BHIS299
BTYR336
BTRP349
BHOH401
BHOH410
EHIS18

site_idAC3
Number of Residues15
DetailsBINDING SITE FOR RESIDUE SAH C 801
ChainResidue
CHOH157
CHOH171
CHOH177
CGLY225
CLYS226
CARG228
CCYS270
CTYR271
CLEU296
CASN298
CHIS299
CTYR336
CTRP349
CHOH363
GHIS18

site_idAC4
Number of Residues18
DetailsBINDING SITE FOR RESIDUE SAH D 801
ChainResidue
BHOH21
DHOH17
DHOH45
DHOH55
DHOH160
DGLY225
DLYS226
DARG228
DCYS270
DTYR271
DARG295
DLEU296
DASN298
DHIS299
DTYR336
DTRP349
EARG23
HHIS18

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues16
DetailsDNA_BIND:
ChainResidueDetails
ELYS16-LYS20
DLYS226
DTYR271
DASN298
FLYS16-LYS20
GLYS16-LYS20
HLYS16-LYS20
BTYR271
BASN298
CLYS226
CTYR271
CASN298

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: N6-propionyllysine; alternate => ECO:0000269|PubMed:17267393
ChainResidueDetails
ELYS16
FLYS16
GLYS16
HLYS16

site_idSWS_FT_FI3
Number of Residues4
DetailsMOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:12086618, ECO:0000269|PubMed:15964846, ECO:0000269|PubMed:17967882, ECO:0000269|PubMed:27338793
ChainResidueDetails
ELYS20
FLYS20
GLYS20
HLYS20

site_idSWS_FT_FI4
Number of Residues8
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2); alternate => ECO:0007744|PubMed:28112733
ChainResidueDetails
ELYS20
FLYS20
GLYS20
HLYS20

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PDB entries from 2024-04-24

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