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3ERT

HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 4-HYDROXYTAMOXIFEN

Replaces:  2ERT
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE OHT A 600
ChainResidue
AHOH2
AGLY521
AHOH58
ALEU346
AALA350
AASP351
AGLU353
ALEU387
AARG394
AMET421

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537

site_idSWS_FT_FI2
Number of Residues1
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447

218853

PDB entries from 2024-04-24

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