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3A2I

Crystal structure of the human vitamin D receptor (H305F) ligand binding domain complexed with TEI-9647

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE TEJ A 1
ChainResidue
ATYR143
APHE305
AHIS397
AVAL234
ASER237
AILE271
AARG274
ASER275
ASER278
ATRP286
AVAL300

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298
ChainResidueDetails
ATYR143
ALEU227
AILE271
APHE305
AHIS397

219515

PDB entries from 2024-05-08

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