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1MRL

Crystal structure of streptogramin A acetyltransferase with dalfopristin

Functional Information from GO Data
ChainGOidnamespacecontents
A0016740molecular_functiontransferase activity
A0016746molecular_functionacyltransferase activity
A0046677biological_processresponse to antibiotic
B0016740molecular_functiontransferase activity
B0016746molecular_functionacyltransferase activity
B0046677biological_processresponse to antibiotic
C0016740molecular_functiontransferase activity
C0016746molecular_functionacyltransferase activity
C0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE DOL A 300
ChainResidue
ATYR54
BTYR37
BASP39
AILE56
AASN81
AHIS82
ALEU93
AMET102
APRO103
ALEU108
BASN14

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE DOL B 301
ChainResidue
ALEU105
AASP106
BTYR54
BASN81
BHIS82
BLEU93
BMET102
BLEU108
CASN14
CVAL17
CTYR37
CASP39

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE DOL C 302
ChainResidue
ATYR37
AASP39
BLYS148
BASN162
CASN81
CHIS82
CLEU93
CMET102
CLEU108

Functional Information from PROSITE/UniProt
site_idPS00101
Number of Residues29
DetailsHEXAPEP_TRANSFERASES Hexapeptide-repeat containing-transferases signature. IGkdVvImpgVkIGdgAiVAanSvVvkdI
ChainResidueDetails
AILE122-ILE150

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE:
ChainResidueDetails
AHIS82
BHIS82
CHIS82

221051

PDB entries from 2024-06-12

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