| PDBID: | 8zmq | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the second bromodomain of human BRD4 BD2 in complex with the inhibitor Y13190 | | Authors: | Li, J., Hu, Q., Xu, H., Zhao, X., Zhang, C., Zhu, R., Wu, X., Zhang, Y., Xu, Y. | | Deposition date: | 2024-05-23 |
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| PDBID: | 8zmb | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of human BRD4 BD1 in complex with the inhibitor Y13195 | | Authors: | Li, J., Hu, Q., Xu, H., Zhao, X., Zhang, C., Zhu, R., Wu, X., Zhang, Y., Xu, Y. | | Deposition date: | 2024-05-22 |
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| PDBID: | 8zm8 | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of human BRD4 BD1 in complex with the inhibitor Y13221 | | Authors: | Li, J., Hu, Q., Xu, H., Zhao, X., Zhang, C., Zhu, R., Wu, X., Zhang, Y., Xu, Y. | | Deposition date: | 2024-05-22 |
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| PDBID: | 9fby | | Status: | HPUB -- hold until publication | | Title: | N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with (5-(4-chloro-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one | | Authors: | Chung, C. | | Deposition date: | 2024-05-14 |
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| PDBID: | 9f1l | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | First bromodomain of BRD4 in complex with ISOX-DUAL based degrader 35 | | Authors: | Balourdas, D.I., Edmonds, A.K., Marsh, G.P., Maple, H.J., Spencer, J., Knapp, S., Joerger, A.C., Structural Genomics Consortium (SGC) | | Deposition date: | 2024-04-19 |
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| PDBID: | 9f1n | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | First bromodomain of BRD4 in complex with ISOX-DUAL based degrader 46 | | Authors: | Balourdas, D.I., Edmonds, A.K., Marsh, G.P., Maple, H.J., Spencer, J., Knapp, S., Joerger, A.C., Structural Genomics Consortium (SGC) | | Deposition date: | 2024-04-19 |
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| PDBID: | 9f1m | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | First bromodomain of BRD4 in complex with ISOX-DUAL based degrader 45 | | Authors: | Balourdas, D.I., Edmonds, A.K., Marsh, G.P., Maple, H.J., Spencer, J., Knapp, S., Joerger, A.C., Structural Genomics Consortium (SGC) | | Deposition date: | 2024-04-19 |
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| PDBID: | 9f1k | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | First bromodomain of BRD4 in complex with ISOX-DUAL based inhibitor 30 | | Authors: | Balourdas, D.I., Edmonds, A.K., Marsh, G.P., Maple, H.J., Spencer, J., Knapp, S., Joerger, A.C., Structural Genomics Consortium (SGC) | | Deposition date: | 2024-04-19 |
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| PDBID: | 9f1j | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | First bromodomain of BRD4 in complex with ISOX-DUAL based degrader 14 | | Authors: | Balourdas, D.I., Edmonds, A.K., Marsh, G.P., Maple, H.J., Spencer, J., Knapp, S., Joerger, A.C., Structural Genomics Consortium (SGC) | | Deposition date: | 2024-04-19 |
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| PDBID: | 8ymb | | Status: | HPUB -- hold until publication | | Title: | The crystal structure of SHD931 in complex with Brd4-BD2 and VCB | | Authors: | Huang, W.X., Chen, Y.H., Li, C.G., Ding, K. | | Deposition date: | 2024-03-08 |
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| PDBID: | 8v9f | | Status: | HPUB -- hold until publication | | Title: | BRD4 BD1 liganded with macrocyclic compound 2d (JJ-II-363A) | | Authors: | Schonbrunn, E., Chan, A. | | Deposition date: | 2023-12-08 | | Sequence: | >Entity 1
SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE
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| PDBID: | 8v92 | | Status: | HPUB -- hold until publication | | Title: | BRD4 BD1 liganded with macrocyclic compound 2b (JJ-II-352A) | | Authors: | Schonbrunn, E., Chan, A. | | Deposition date: | 2023-12-07 | | Sequence: | >Entity 1
SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE
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| PDBID: | 8wqo | | Status: | AUTH -- processed, waiting for author review and approval | | Title: | Crystal structure of BRD4-BD1 bound with DI106 | | Authors: | Cao, D., Xiong, B. | | Deposition date: | 2023-10-12 |
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| PDBID: | 8qal | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of BRD4 in complex with acetyl-pyrrole derivative compound 83 | | Authors: | Dalle Vedove, A., Cazzanelli, G., Lolli, G. | | Deposition date: | 2023-08-23 |
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| PDBID: | 8qan | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of BRD4 in complex with acetyl-pyrrole derivative compound 79 | | Authors: | Dalle Vedove, A., Cazzanelli, G., Lolli, G. | | Deposition date: | 2023-08-23 |
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| PDBID: | 8qap | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of BRD4 in complex with acetyl-pyrrole derivative compound 2 | | Authors: | Dalle Vedove, A., Cazzanelli, G., Lolli, G. | | Deposition date: | 2023-08-23 |
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| PDBID: | 8qar | | Status: | HPUB -- hold until publication | | Title: | Crystal Structure of the first bromodomain of BRD4 in complex with acetyl-pyrrole derivative compound 98 | | Authors: | Dalle Vedove, A., Cazzanelli, G., Lolli, G. | | Deposition date: | 2023-08-23 |
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| PDBID: | 8htl | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal structure of BRD4-BD1 bound with DI106 | | Authors: | Cao, D., Xiong, B. | | Deposition date: | 2022-12-21 |
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| PDBID: | 7zfq | | Status: | WDRN -- deposition withdrawn | | Title: | BRD4 in complex with FragLite29 | | Authors: | Turberville, S., Martin, M.P., Hope, I., Noble, M.E.M. | | Deposition date: | 2022-04-01 |
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| PDBID: | 7lwx | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal structure of BRD4 bromodomain 1 with 1-(2-methyl-4-phenoxy-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)indolin-1-yl)ethan-1-one | | Authors: | Ilyichova, O.V., Jennings, I.G., Scanlon, M.J., Thompson, P.E. | | Deposition date: | 2021-03-02 |
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| PDBID: | 5zip | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal Structure of the first bromodomain of human BRD4 in complex with 5-((4-fluoro-1H-imidazol-1-yl)methyl)quinolin-8-ol | | Authors: | Xing, J., Zhang, R.K., Zheng, M.Y., Luo, C., Jiang, X.R. | | Deposition date: | 2018-03-16 | | Release date: | 2019-04-20 |
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| PDBID: | 5jc2 | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal structure of Brd4 bromodomain 1 with compound 3 | | Authors: | Broadbeck, D., Gill, A., Hafenbradl, D., Hartley, D., Hubbard, P., Lock, C., Ritchie, A., Sheppard, D.W., MacLeod, A.M. | | Deposition date: | 2016-04-14 |
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| PDBID: | 5jc4 | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal structure of Brd4 bromodomain 1 with compound 15 | | Authors: | Broadbeck, D., Gill, A., Hafenbradl, D., Hartley, D., Hubbard, P., Lock, C., Ritchie, A., Sheppard, D.W., MacLeod, A.M. | | Deposition date: | 2016-04-14 |
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| PDBID: | 5egx | | Status: | WDRN -- deposition withdrawn | | Title: | FIRST DOMAIN OF HUMAN BROMODOMAIN BRD4 IN COMPLEXE WITH INHIBITOR 8-(5-Amino-1H-[1,2,4]triazol-3-ylsulfanylmethyl)-3-(4-chlorobenzyl)-7-ethyl-3,7-dihydropurine-2,6-dione | | Authors: | Raux, B., Rebuffet, E., Betzi, S., Morelli, X. | | Deposition date: | 2015-10-27 |
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| PDBID: | 5e87 | | Status: | WDRN -- deposition withdrawn | | Title: | Crystal structure of the first bromodomain of human BRD4 in complex with MS402 | | Authors: | Plotnikov, A.N., Joshua, j., Zhou, M.-M. | | Deposition date: | 2015-10-13 |
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