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1BK9
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PHOSPHOLIPASE A2 MODIFIED BY PBPB
分子名称: 1,4-BUTANEDIOL, CALCIUM ION, PHOSPHOLIPASE A2, ...
著者Zhao, H, Tang, L, Wang, X, Lin, Z, Zhou, Y.
登録日1998-07-16
公開日1999-03-02
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of a snake venom phospholipase A2 modified by p-bromo-phenacyl-bromide.
Toxicon, 36, 1998
1BVM
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SOLUTION NMR STRUCTURE OF BOVINE PANCREATIC PHOSPHOLIPASE A2, 20 STRUCTURES
分子名称: PROTEIN (PHOSPHOLIPASE A2)
著者Yuan, C.-H, Byeon, I.-J.L, Li, Y, Tsai, M.-D.
登録日1998-09-14
公開日1999-09-16
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Structural analysis of phospholipase A2 from functional perspective. 1. Functionally relevant solution structure and roles of the hydrogen-bonding network.
Biochemistry, 38, 1999
1B4W
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BASIC PHOSPHOLIPASE A2 FROM AGKISTRODON HALYS PALLAS-IMPLICATIONS FOR ITS ASSOCIATION AND ANTICOAGULANT ACTIVITIES BY X-RAY CRYSTALLOGRAPHY
分子名称: PROTEIN (PHOSPHOLIPASE A2), octyl beta-D-glucopyranoside
著者Zhao, K.H, Lin, Z.J.
登録日1998-12-30
公開日2000-01-12
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure of basic phospholipase A2 from Agkistrodon halys Pallas: implications for its association, hemolytic and anticoagulant activities.
Toxicon, 38, 2000
1GOD
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MONOMERIC LYS-49 PHOSPHOLIPASE A2 HOMOLOGUE ISOLATED FROM THE VENOM OF CERROPHIDION (BOTHROPS) GODMANI
分子名称: PROTEIN (PHOSPHOLIPASE A2)
著者Arni, R.K, Fontes, M.R.M, Barberato, C, Gutierrez, J.M, Diaz-Oreiro, C, Ward, R.J.
登録日1999-04-16
公開日1999-04-23
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of myotoxin II, a monomeric Lys49-phospholipase A2 homologue isolated from the venom of Cerrophidion (Bothrops) godmani.
Arch.Biochem.Biophys., 366, 1999
1CL5
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CRYSTAL STRUCTURE OF PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA
分子名称: PROTEIN (PHOSPHOLIPASE A2)
著者Chandra, V, Kaur, P, Singh, T.P.
登録日1999-05-06
公開日1999-05-12
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Three-dimensional structure of a presynaptic neurotoxic phospholipase A2 from Daboia russelli pulchella at 2.4 A resolution.
J.Mol.Biol., 296, 2000
1C1J
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STRUCTURE OF CADMIUM-SUBSTITUTED PHOSPHOLIPASE A2 FROM AGKISTRONDON HALYS PALLAS AT 2.8 ANGSTROMS RESOLUTION
分子名称: BASIC PHOSPHOLIPASE A2, CADMIUM ION, octyl beta-D-glucopyranoside
著者Zhang, H.-l, Zhang, Y.-q, Song, S.-y, Zhou, Y, Lin, Z.-j.
登録日1999-07-22
公開日2002-07-05
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of Cadmium-substituted Phospholipase A2 from Agkistrodon halys Pallas at 2.8 Angstroms Resolution
Protein Pept.Lett., 6, 1999
1QLL
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Piratoxin-II (Prtx-II) - a K49 PLA2 from Bothrops pirajai
分子名称: N-TRIDECANOIC ACID, PHOSPHOLIPASE A2
著者Lee, W.-H, Polikarpov, I.
登録日1999-09-01
公開日2000-09-07
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Structural Basis for Low Catalytic Activity in Lys49 Phospholipases A2-A Hypothesis: The Crystal Structure of Piratoxin II Complexed to Fatty Acid
Biochemistry, 40, 2001
1DB5
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HUMAN S-PLA2 IN COMPLEX WITH INDOLE 6
分子名称: 4-(1-BENZYL-3-CARBAMOYLMETHYL-2-METHYL-1H-INDOL-5-YLOXY)-BUTYRIC ACID, CALCIUM ION, PROTEIN (PHOSPHOLIPASE A2)
著者Chirgadze, N.Y, Schevitz, R.W, Wery, J.-P.
登録日1999-11-02
公開日1999-11-12
最終更新日2012-02-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure-based design of the first potent and selective inhibitor of human non-pancreatic secretory phospholipase A2.
Nat.Struct.Biol., 2, 1995
1DB4
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HUMAN S-PLA2 IN COMPLEX WITH INDOLE 8
分子名称: CALCIUM ION, PHOSPHOLIPASE A2, [3-(1-BENZYL-3-CARBAMOYLMETHYL-2-METHYL-1H-INDOL-5-YLOXY)-PROPYL-]-PHOSPHONIC ACID
著者Chirgadze, N.Y, Schevitz, R.W, Wery, J.-P.
登録日1999-11-02
公開日1999-11-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure-based design of the first potent and selective inhibitor of human non-pancreatic secretory phospholipase A2.
Nat.Struct.Biol., 2, 1995
1DCY
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CRYSTAL STRUCTURE OF HUMAN S-PLA2 IN COMPLEX WITH INDOLE 3 ACTIVE SITE INHIBITOR
分子名称: 1-BENZYL-5-METHOXY-2-METHYL-1H-INDOL-3-YL)-ACETIC ACID, CALCIUM ION, PHOSPHOLIPASE A2
著者Chirgadze, N.Y, Schevitz, R.W, Wery, J.-P.
登録日1999-11-05
公開日1999-11-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure-based design of the first potent and selective inhibitor of human non-pancreatic secretory phospholipase A2.
Nat.Struct.Biol., 2, 1995
1DPY
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THREE-DIMENSIONAL STRUCTURE OF A NOVEL PHOSPHOLIPASE A2 FROM INDIAN COMMON KRAIT AT 2.45 A RESOLUTION
分子名称: PHOSPHOLIPASE A2, SODIUM ION
著者Singh, G, Gourinath, S, Sharma, S, Paramasivam, M, Srinivasan, A, Singh, T.P.
登録日1999-12-28
公開日2000-06-28
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Sequence and crystal structure determination of a basic phospholipase A2 from common krait (Bungarus caeruleus) at 2.4 A resolution: identification and characterization of its pharmacological sites.
J.Mol.Biol., 307, 2001
1C74
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Structure of the double mutant (K53,56M) of phospholipase A2
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Sekar, K, Tsai, M.D, Jain, M.K, Ramakumar, S.
登録日2000-01-22
公開日2000-07-22
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural basis of the anionic interface preference and k*cat activation of pancreatic phospholipase A2.
Biochemistry, 39, 2000
1FB2
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STRUCTURE OF PHOSPHOLIPASE A2 FROM DABOIA RUSSELLI PULCHELLA AT 1.95
分子名称: PHOSPHOLIPASE A2
著者Chandra, V, Kaur, P, Betzel, C, Singh, T.P.
登録日2000-07-14
公開日2001-07-25
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Regulation of catalytic function by molecular association: structure of phospholipase A2 from Daboia russelli pulchella (DPLA2) at 1.9 A resolution.
Acta Crystallogr.,Sect.D, 57, 2001
1FE5
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SEQUENCE AND CRYSTAL STRUCTURE OF A BASIC PHOSPHOLIPASE A2 FROM COMMON KRAIT (BUNGARUS CAERULEUS) AT 2.4 RESOLUTION: IDENTIFICATION AND CHARACTERIZATION OF ITS PHARMACOLOGICAL SITES.
分子名称: CALCIUM ION, PHOSPHOLIPASE A2
著者Singh, G, Gourinath, S, Sharma, S, Paramasivam, M, Srinivasan, A, Singh, T.P.
登録日2000-07-21
公開日2001-01-24
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Sequence and crystal structure determination of a basic phospholipase A2 from common krait (Bungarus caeruleus) at 2.4 A resolution: identification and characterization of its pharmacological sites.
J.Mol.Biol., 307, 2001
1FV0
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FIRST STRUCTURAL EVIDENCE OF THE INHIBITION OF PHOSPHOLIPASE A2 BY ARISTOLOCHIC ACID: CRYSTAL STRUCTURE OF A COMPLEX FORMED BETWEEN PHOSPHOLIPASE A2 AND ARISTOLOCHIC ACID
分子名称: 1,4-DIETHYLENE DIOXIDE, 9-HYDROXY ARISTOLOCHIC ACID, ACETATE ION, ...
著者Chandra, V, Jasti, J, Kaur, P, Srinivasan, A, Betzel, C, Singh, T.P.
登録日2000-09-18
公開日2002-08-28
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Basis of Phospholipase A2 Inhibition for the Synthesis of Prostaglandins by the Plant Alkaloid Aristolochic Acid from a 1.7 A Crystal Structure
Biochemistry, 41, 2002
1FX9
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CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + SULPHATE IONS)
分子名称: 1-HEXADECYL-3-TRIFLUOROETHYL-SN-GLYCERO-2-PHOSPHATE METHANE, CALCIUM ION, PHOSPHOLIPASE A2, ...
著者Pan, Y.H, Epstein, T.M, Jain, M.K, Bahnson, B.J.
登録日2000-09-25
公開日2001-09-25
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Five coplanar anion binding sites on one face of phospholipase A2: relationship to interface binding.
Biochemistry, 40, 2001
1FXF
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CARBOXYLIC ESTER HYDROLASE COMPLEX (DIMERIC PLA2 + MJ33 INHIBITOR + PHOSPHATE IONS)
分子名称: 1-HEXADECYL-3-TRIFLUOROETHYL-SN-GLYCERO-2-PHOSPHATE METHANE, CALCIUM ION, PHOSPHATE ION, ...
著者Pan, Y.H, Epstein, T.M, Jain, M.K, Bahnson, B.J.
登録日2000-09-25
公開日2001-09-25
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Five coplanar anion binding sites on one face of phospholipase A2: relationship to interface binding.
Biochemistry, 40, 2001
1G0Z
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SPECIFIC MUTATIONS IN KRAIT PLA2 LEAD TO DIMERIZATION OF PROTEIN MOLECULES: CRYSTAL STRUCTURE OF KRAIT PLA2 AT 2.1 RESOLUTION
分子名称: CHLORIDE ION, PHOSPHOLIPASE A2
著者Singh, T.P, Gourinath, S, Sharma, S, Singh, G.
登録日2000-10-10
公開日2003-06-17
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Specific mutations in Krait PLA2 lead to dimerization of protein molecules: Crystal structure of Krait PLA2 at 2.1 resolution.
To be Published
1G2X
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Sequence induced trimerization of krait PLA2: crystal structure of the trimeric form of krait PLA2
分子名称: PHOSPHOLIPASE A2
著者Singh, G, Gourinath, S, Sharma, S, Bhanumathi, S, Paramsivam, M, Singh, T.P.
登録日2000-10-22
公開日2003-06-17
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Sequence-induced trimerization of phospholipase A2: structure of a trimeric isoform of PLA2 from common krait (Bungarus caeruleus) at 2.5 A resolution.
Acta Crystallogr.,Sect.F, 61, 2005
1G4I
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Crystal structure of the bovine pancreatic phospholipase A2 at 0.97A
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, ...
著者Steiner, R.A, Rozeboom, H.J, de Vries, A, Kalk, K.H, Murshudov, G.N, Wilson, K.S, Dijkstra, B.W.
登録日2000-10-27
公開日2001-04-04
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (0.97 Å)
主引用文献X-ray structure of bovine pancreatic phospholipase A2 at atomic resolution.
Acta Crystallogr.,Sect.D, 57, 2001
1GH4
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Structure of the triple mutant (K56M, K120M, K121M) of phospholipase A2
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, PHOSPHOLIPASE A2
著者Sekar, K, Velmurugan, D, Tsai, M.D.
登録日2000-11-09
公開日2001-05-09
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Observation of additional calcium ion in the crystal structure of the triple mutant K56,120,121M of bovine pancreatic phospholipase A2.
J.Mol.Biol., 324, 2002
1HN4
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PROPHOSPHOLIPASE A2 DIMER COMPLEXED WITH MJ33, SULFATE, AND CALCIUM
分子名称: 1-HEXADECYL-3-TRIFLUOROETHYL-SN-GLYCERO-2-PHOSPHATE METHANE, CALCIUM ION, PROPHOSPHOLIPASE A2, ...
著者Epstein, T.M, Pan, Y.H, Jain, M.K, Bahnson, B.J.
登録日2000-12-06
公開日2001-12-05
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The basis for k(cat) impairment in prophospholipase A(2) from the anion-assisted dimer structure.
Biochemistry, 40, 2001
1IJL
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Crystal structure of acidic phospholipase A2 from deinagkistrodon acutus
分子名称: CALCIUM ION, PHOSPHOLIPASE A2, ZINC ION
著者Gu, L, Zhang, H, Song, S, Zhou, Y, Lin, Z.
登録日2001-04-27
公開日2001-12-28
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure of an acidic phospholipase A2 from the venom of Deinagkistrodon acutus.
Acta Crystallogr.,Sect.D, 58, 2002
1JLT
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Vipoxin Complex
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, PHOSPHOLIPASE A2, ...
著者Banumathi, S, Rajashankar, K.R, Notzel, C, Aleksiev, B, Singh, T.P, Genov, N, Betzel, C.
登録日2001-07-16
公開日2001-10-31
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structure of the neurotoxic complex vipoxin at 1.4 A resolution.
Acta Crystallogr.,Sect.D, 57, 2001
1JQ8
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Design of specific inhibitors of phospholipase A2: Crystal structure of a complex formed between phospholipase A2 from Daboia russelli pulchella and a designed pentapeptide Leu-Ala-Ile-Tyr-Ser at 2.0 resolution
分子名称: ACETIC ACID, Peptide inhibitor, Phospholipase A2, ...
著者Chandra, V, Jasti, J, Kaur, P, Dey, S, Betzel, C, Singh, T.P.
登録日2001-08-04
公開日2002-11-06
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Design of specific peptide inhibitors of phospholipase A2: structure of a complex formed between Russell's viper phospholipase A2 and a designed peptide Leu-Ala-Ile-Tyr-Ser (LAIYS).
ACTA CRYSTALLOGR.,SECT.D, 58, 2002

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