3BJQ
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![BU of 3bjq by Molmil](/molmil-images/mine/3bjq) | |
4O81
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![BU of 4o81 by Molmil](/molmil-images/mine/4o81) | |
4OE9
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![BU of 4oe9 by Molmil](/molmil-images/mine/4oe9) | |
3BDV
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![BU of 3bdv by Molmil](/molmil-images/mine/3bdv) | |
3BF4
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![BU of 3bf4 by Molmil](/molmil-images/mine/3bf4) | |
3C26
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![BU of 3c26 by Molmil](/molmil-images/mine/3c26) | |
3BJX
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3BKX
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![BU of 3bkx by Molmil](/molmil-images/mine/3bkx) | |
4LQX
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![BU of 4lqx by Molmil](/molmil-images/mine/4lqx) | |
3BWV
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![BU of 3bwv by Molmil](/molmil-images/mine/3bwv) | |
3C8U
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![BU of 3c8u by Molmil](/molmil-images/mine/3c8u) | |
3BY7
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![BU of 3by7 by Molmil](/molmil-images/mine/3by7) | |
3C18
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![BU of 3c18 by Molmil](/molmil-images/mine/3c18) | |
4MRU
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![BU of 4mru by Molmil](/molmil-images/mine/4mru) | |
3C3P
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3BLN
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3WYX
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![BU of 3wyx by Molmil](/molmil-images/mine/3wyx) | CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH 6-((3-(cyanomethoxy)-4-(1-methyl-1H-pyrazol-4-yl)phenyl)amino)-2-(cyclohexylamino)nicotinonitrile | Descriptor: | 6-{[3-(cyanomethoxy)-4-(1-methyl-1H-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile, Dual specificity protein kinase TTK, IODIDE ION | Authors: | Kusakabe, K, Ide, N, Daigo, Y, Itoh, T, Yamamoto, T, Kojima, E, Mitsuoka, Y, Tadano, G, Tagashira, S, Higashino, K, Okano, Y, Sato, Y, Inoue, M, Iguchi, M, Kanazawa, T, Ishioka, Y, Dohi, K, Kido, Y, Sakamoto, S, Ando, S, Maeda, M, Higaki, M, Yoshizawa, H, Mura, H, Nakamura, Y. | Deposit date: | 2014-09-09 | Release date: | 2015-04-08 | Last modified: | 2024-05-29 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | A unique hinge binder of extremely selective aminopyridine-based Mps1 (TTK) kinase inhibitors with cellular activity. Bioorg.Med.Chem., 23, 2015
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4RVO
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3BXP
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![BU of 3bxp by Molmil](/molmil-images/mine/3bxp) | |
3C6C
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3C8L
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3BWX
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![BU of 3bwx by Molmil](/molmil-images/mine/3bwx) | |
3BN7
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4OHQ
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![BU of 4ohq by Molmil](/molmil-images/mine/4ohq) | |
3V43
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![BU of 3v43 by Molmil](/molmil-images/mine/3v43) | Crystal structure of MOZ | Descriptor: | ACETATE ION, Histone H3.1, Histone acetyltransferase KAT6A, ... | Authors: | Qiu, Y, Li, F. | Deposit date: | 2011-12-14 | Release date: | 2012-06-27 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Combinatorial readout of unmodified H3R2 and acetylated H3K14 by the tandem PHD finger of MOZ reveals a regulatory mechanism for HOXA9 transcription Genes Dev., 26, 2012
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