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PDB: 5 results

2WUH
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BU of 2wuh by Molmil
Crystal structure of the DDR2 discoidin domain bound to a triple- helical collagen peptide
Descriptor: COLLAGEN PEPTIDE, DISCOIDIN DOMAIN RECEPTOR 2
Authors:Carafoli, F, Bihan, D, Stathopoulos, S, Konitsiotis, A.D, Kvansakul, M, Farndale, R.W, Leitinger, B, Hohenester, E.
Deposit date:2009-10-05
Release date:2009-12-29
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Crystallographic Insight Into Collagen Recognition by Discoidin Domain Receptor 2
Structure, 17, 2009
7AYM
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BU of 7aym by Molmil
Structure of DDR2 Kinase domain in complex with IBZ3
Descriptor: Discoidin domain-containing receptor 2,Epithelial discoidin domain-containing receptor 1, N-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide
Authors:Nawrotek, A, Talagas, A, Vuillard, L.M, Miallau, L.
Deposit date:2020-11-12
Release date:2020-12-16
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.12 Å)
Cite:Structure of DDR2 Kinase domain in complex with IBZ3
To Be Published
7AZB
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BU of 7azb by Molmil
Structure of DDR2 DS domain in complex with VHH
Descriptor: Discoidin domain-containing receptor 2, VHH
Authors:Talagas, A, Nawrotek, A, Arrial, A, Vuillard, L.M, Miallau, L.
Deposit date:2020-11-16
Release date:2020-11-25
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.62 Å)
Cite:Structure of DDR2 DS domain in complex with VHH
To Be Published
6FER
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BU of 6fer by Molmil
Crystal Structure of human DDR2 kinase in complex with 2-[4,5-difluoro-2-oxo-1'-(1H-pyrazolo[3,4-b]pyridine-5-carbonyl)spiro[indole-3,4'-piperidine]-1-yl]-N-(2,2,2-trifluoroethyl)acetamide
Descriptor: 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{H}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{N}-[2,2,2-tris(fluoranyl)ethyl]ethanamide, Discoidin domain-containing receptor 2
Authors:Stihle, M, Richter, H, Benz, J, Kuhn, B, Rudolph, M.G.
Deposit date:2018-01-03
Release date:2018-11-28
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.87 Å)
Cite:DNA-Encoded Library-Derived DDR1 Inhibitor Prevents Fibrosis and Renal Function Loss in a Genetic Mouse Model of Alport Syndrome.
Acs Chem.Biol., 14, 2019
2Z4F
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BU of 2z4f by Molmil
Solution structure of the Discoidin Domain of DDR2
Descriptor: Discoidin domain-containing receptor 2
Authors:Ichikawa, O, Osawa, M, Nishida, N, Goshima, N, Nomura, N, Shimada, I.
Deposit date:2007-06-16
Release date:2007-09-04
Last modified:2022-03-16
Method:SOLUTION NMR
Cite:Structural basis of the collagen-binding mode of discoidin domain receptor 2
Embo J., 26, 2007

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